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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0865 | Ranitidine Hydrochloride | AH19065 | P450 , Antibacterial , Histamine Receptor |
Ranitidine Hydrochloride (AH19065) is a member of the class of histamine H2-receptor antagonists with antacid activity. Ranitidine is a competitive and reversible inhibitor of the action of histamine, released by enteroc... | |||
T3610 | Ranitidine | HSDB 3925,Ranitidin | P450 , Antibacterial , Histamine Receptor |
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers. | |||
T7524 | Metiamide | SK&F 92058 | Histamine Receptor |
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist . | |||
T15195 | Ebrotidine | FI3542 | Histamine Receptor |
Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection. | |||
T0157 | Roxatidine Acetate hydrochloride | HOE 760,Roxatidine Acetate HCl | Histamine Receptor |
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation. | |||
T1575 | Nizatidine | Axid,Acinon,Zanizal | AChE , Histamine Receptor |
Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity. | |||
T31195 | Dalcotidine | KU 1257,KU-1257 | Histamine Receptor |
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value f... | |||
T68146 | Sufotidine | AH 25352X,AH25352X,AH-25352X | Histamine Receptor |
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist. | |||
T68056 | Donetidine | Histamine Receptor | |
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders. | |||
T68122L | Oxmetidine FA | Oxmetidine FA(72830-39-8 Free base) | Histamine Receptor |
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties. | |||
T8599 | Betazole dihydrochloride | Betazole hydrochloride | Histamine Receptor |
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor. | |||
T22842 | HTMT dimaleate | Histamine Trifluoromethyl Toluidide Dimaleate | Histamine Receptor |
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist. | |||
T68921 | Impromidine hydrochloride | Histamine Receptor | |
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies. | |||
T1627 | Famotidine | MK-208 | Histamine Receptor |
Famotidine (MK-208) is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors located on the basolateral membrane of the parietal cell, famotidi... | |||
T15005 | CP-66948 | Histamine Receptor | |
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa. | |||
T11825 | LCB-2853 | PPAR | |
LCB-2853 is a potent thromboxane A2/prostaglandin H2 (TXA2/PGH2) receptor antagonist with antiplatelet aggregation, antivasospasm, and antithrombotic effects. | |||
T68100 | Mifentidine | DA 4577 | Histamine Receptor |
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers. | |||
T22724 | Dimaprit dihydrochloride | NOS , NO Synthase , Histamine Receptor | |
Dimaprit dihydrochloride is a selective histamine H2 receptor agonist. Dimaprit dihydrochloride also inhibits nNOS with an IC50 of 49 μM. It can stimulate gastric acid secretion. | |||
T10000 | (±)-Tazifylline | Histamine Receptor | |
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptors, 5-hydroxytryptamine and muscarinic receptor subtypes. | |||
T68122 | Oxmetidine | SKF 92994,Oxmetidina,Oxmetidinum | Histamine Receptor |
Oxmetidine (SKF 92994) is a novel H2 receptor antagonist that is cytotoxic. Oxmetidine inhibits transmembrane calcium flux in cardiac and vascular tissues and is used in the treatment of active duodenal ulcers. |