Home Tools
Log in
Cart

Search Result

Search Results for " gpr35 "

17

Compounds

Cat No. Product Name Synonyms Targets
T23434 GPR35 agonist 2 TC-G 1001 GPR , Arrestin
GPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist 2 in the β-arrestin and Ca2+ release assays were 26 and 3.2 nM, respectively.
T11455 GPR35 agonist 1 Others
GPR35 agonist 1 is a highly effective and specific GPR35/CXCR8 agonist (EC50: 5.8 nM).
T72755 GPR35 agonist 3
GPR35 agonist 3, a synthetic compound, acts as an agonist for GPR35 with an EC50 value of 1.4 μM and is utilized in researching numerous diseases including gastric cancer, type 2 diabetes, cardiovascular diseases, and di...
T9162 CID1231538 GPR
CID1231538 is a potent GPR35 antagonist.
T21874 CID 2745687 GPR
CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn disodium and zaprinast, two agonists that share an overlapping binding site.
T21622 Tyrphostin A25 AG-82,Tyrphostin AG 82,RG-50875 EGFR , GPR
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.
T2129 Zaprinast PDE
Zaprinast is a cGMP-selective phosphodiesterase (PDE) inhibitor and a GPR35 agonist. It has a strong activating effect on rat GPR35 and a certain activating effect on human GPR35. It reduces vascular remodeling through a...
T22103 ML-193 CID 1261822 Cannabinoid Receptor
ML-193 (CID 1261822) is a potent and selective GPR55 antagonist( IC50 : 221 nM). It shows more than 27-fold selectivity for GPR55 over GPR35, CB1 and CB2, and can improve the motor and the sensorimotor deficits of Parkin...
T65135 Kynurenic acid Fibrostop 2,Quinurenic acid GPR , GluR , NMDAR
Kynurenic acid (Quinurenic acid) is an endogenous tryptophan active metabolite, a triple antagonist of NMDA, glutamate, α7 nicotinic acetylcholine receptor, and an agonist of GPR35/CXCR8 with neuroprotective and anticonv...
T8571 ML-184 CID2440433 Cannabinoid Receptor
ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.
T23120 Pamoic acid disodium Pamoic acid disodium salt Others
Pamoic acid disodium is a GPR35 agonist.
T22158 TCS 3035
GPR35 agonist 4 (compound 10) serves as a potent GPR35 agonist, showcasing a pEC50 of 5.86, indicating its high potency towards both human and rat GPR35. Notably, the mutation of arginine at position 3.36 results in the ...
T23542 YE 120 Others
YE 120 is a GPR35 agonist.
T12074 ML 145 Others
ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)
T73665 Bufrolin
Bufrolin, an analog of Cromoglycate (histamine release inhibitor) and a potent agonist of GPR35, enhances the interaction between β-arrestin-2 and both human GPR35a and rat GPR35. It stabilizes mast cells, exhibiting ant...
TQ0075 ML314 Neurotensin Receptor
ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased neurotensin receptor ligand for methamphetamine abuse that inhibits NTR2 and GPR35.
T37529 TC NTR1 17
Non-peptide neurotensin receptor 1 (NTS1) partial agonist (EC50 <15.6 nM and Emax = 63% of neurotensin response in Ca2+ mobilization assay). Exhibits over 50-fold selectivity for NTS1 over NTS2 and GPR35. Hershberger et ...
TargetMol