20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T76566 | Fsh receptor-binding inhibitor fragment(bi-10) | ||
FSH receptor-binding inhibitor fragment (bi-10) is a potent antagonist that inhibits the binding of follicle-stimulating hormone (FSH) to its receptor (FSHR), modifying FSH activity at the receptor level. It suppresses o... | |||
T1908 | MHY1485 | mTOR , Autophagy | |
MHY1485 is a mTOR activator. It inhibits the autophagic process by inhibition of fusion between autophagosomes and lysosomes, leading to the accumulation of LC3II protein and enlarged autophagosomes. | |||
T3630 | Relugolix | RVT-601,TAK-385 | GNRH Receptor |
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively bi... | |||
T21308 | Histrelin | Supprelin LA,Histrelin Acetate | Others |
Histrelin (Supprelin LA) acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It is considered a GnRH agonist. Histrelin is used in the treatment of hormone-sensitive cancers of th... | |||
T76222 | HFSH-β-(33-53) (TFA) | ||
hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist. It prevents FSH from binding to its receptor and partially p... | |||
T72835 | FSHR agonist 1 | ||
FSHR agonist 1, an allosteric agonist of the follicle-stimulating hormone receptor (FSHR), exhibits high affinity, with a pEC50 of 7.72. It forms extensive interactions with the transmembrane domain (TMD) to directly act... | |||
T9380L | Antide acetate | Antide acetate (112568-12-4 Free base) | LHRH |
Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. | |||
TP1342L | GnRH-I acetate | GnRH-I acetate(33515-09-2 free base) | Others |
GnRH-I acetate in release of biologically active Follicle-Stimulating Hormone (FSH) and Luteinizing Hormone (LH) in the blood. | |||
T5520L | Cetrorelix diacetate | NS-75A,SB-075 acetate,SB-075 diacetate,Cetrorelix acetate,NS-75A diacetate | GNRH Receptor |
Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) ... | |||
T21309 | Nafarelin acetate(76932-56-4 free base) | RS-94991-298,Nafarelin acetate,Nafarelin acetate hydrate,Synarel | GNRH Receptor |
Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing h... | |||
T2597 | Norgestrel | SH-850,FH 122-A,WY-3707,SH-70850 | Estrogen/progestogen Receptor , Reactive Oxygen Species |
Norgestrel (WY-3707) is a synthetic progestin commonly used alone or in combination with an estrogen for contraception. Norgestrel suppresses the secretion of luteinizing and follicle-stimulating hormones (LH and FSH), t... | |||
T21410 | Triptorelin acetate(57773-63-4 free base) | Wy 42422,Triptorelin Acetate,CL 118532,AY 25650,CL 118,532,Wy 42462,BIM 21003 | GNRH Receptor |
Triptorelin acetate(57773-63-4 free base) (CL 118,532) is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) by causing constant stim... | |||
T2S2108 | Coixol | 6-methoxybenzoxazolone,6-MBOA,6-Methoxy-2-benzoxazolinone,MBOA | Others , Antibacterial |
1. Coixol (MBOA) acts as a central muscle relaxant with an anti-convulsant effect. 2. Coixol interacts with the pituitary to stimulate reproduction in voles. 3. Coixol has the ability to interact with FSH to stimulate fo... | |||
T25443 | FW 34569 | FW-34-569,FW34569,FW 34-569,FW-34569,FW34-569 | |
FW 34569 is an enkephalin analogue. It stimulated growth hormones and prolactin release and inhibited the release of cortisol and LH, while FSH remained unchanged. | |||
T83489 | [Lys8] LH-RH | ||
[Lys8] LH-RH, an analogue of LH-RH, effectively stimulates the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) [1]. | |||
T82162 | Human follicular gonadotropin releasing peptide | hF-GRP | |
Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH) and follicle-stimulating hormone (FSH) [1] [2]. | |||
T82307 | Glp-His-Pro-Gly-NH2 | pGlu-His-Pro-Gly-NH2 | |
pGlu-His-Pro-Gly-NH2, also known as Glp-His-Pro-Gly-NH2, is a tetrapeptide that promotes the release of gonadotropin, luteinizing hormone (LH), and follicle-stimulating hormone (FSH) [1] [2]. | |||
T83498 | [D-Phe2,D-Ala6]-LH-RH | Wy 18185 | |
[D-Phe2,D-Ala6]-LH-RH is a potent luteinizing hormone-releasing hormone (LH-RH) antagonist with demonstrated activities against LH/FSH-RH and an ability to inhibit ovulation [1]. | |||
T78515 | Follicle-stimulating hormone | Others | |
Follicle-stimulating hormone (FSH), a heterodimeric glycoprotein synthesized by gonadotrophs in the anterior pituitary gland, influences animal fertility and reproductive performance [1] [2]. | |||
T70309 | Dicetrorelix pamoate | ||
Dicetrorelix pamoate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH)... |