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Cetrorelix diacetate

Catalog No. T5520L CAS 130143-01-0

Synonyms: NS-75A, SB-075 acetate, SB-075 diacetate, Cetrorelix acetate, NS-75A diacetate

Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) and follicle-stimulating hormone (FSH).

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Cetrorelix diacetate, CAS 130143-01-0

Pack Size	Availability	Price/USD
1 mg	In stock	$ 48.00
5 mg	In stock	$ 92.00
10 mg	In stock	$ 153.00
25 mg	In stock	$ 307.00
50 mg	In stock	$ 460.00
100 mg	In stock	$ 676.00
500 mg	In stock	$ 1,430.00
1 mL * 10 mM (in DMSO)	In stock	$ 265.00

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Purity: 98.38%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	NS-75A, SB-075 acetate, SB-075 diacetate, Cetrorelix acetate, NS-75A diacetate
Molecular Weight	1551.17
Formula	C74H100ClN17O18
CAS No.	130143-01-0

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (33.53 mM), Sonification is recommended.

H2O: 2 mg/mL (1.34 mM), Sonification is recommended.

References and Literature

1. Tur-Kaspa I, Ezcurra D. GnRH antagonist, cetrorelix, for pituitary suppression in modern, patient-friendly assisted reproductive technology. Expert Opin Drug Metab Toxicol. 2009 Oct;5(10):1323-36. doi: 10.1517/17425250903279969. Review. PubMed PMID: 19761413. 2. Finas D, Hornung D, Diedrich K, Schultze-Mosgau A. Cetrorelix in the treatment of female infertility and endometriosis. Expert Opin Pharmacother. 2006 Oct;7(15):2155-68. Review. PubMed PMID: 17020439. 3. Reissmann T, Schally AV, Bouchard P, Riethmiiller H, Engel J. The LHRH antagonist cetrorelix: a review. Hum Reprod Update. 2000 Jul-Aug;6(4):322-31. Review. PubMed PMID: 10972520. 4. Griesinger G, Felberbaum RE, Schultze-Mosgau A, Diedrich K. Gonadotropin-releasing hormone antagonists for assisted reproductive techniques: are there clinical differences between agents? Drugs. 2004;64(6):563-75. Review. PubMed PMID: 15018588.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Approved Drug Library Anti-Cancer Drug Library Peptide Compound Library NO PAINS Compound Library Bioactive Compound Library Inhibitor Library Bioactive Compounds Library Max Anti-Cancer Compound Library GPCR Compound Library Drug Repurposing Compound Library

Related Products

Related compounds with same targets

Abarelix Linzagolix Deslorelin acetate(57773-65-6 free base) Elagolix sodium Triptorelin acetate(57773-63-4 free base) Ganirelix Acetate Buserelin Acetate (57982-77-1 free base) LGnRH-III, lamprey acetate(147859-97-0 free base)

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Cetrorelix diacetate 130143-01-0 GPCR/G Protein GNRH Receptor SB 075 Diacetate GNRHR SB075 Acetate inhibit GnRH Receptor NS-75A NS-75A Diacetate SB-075 Acetate SB075 Diacetate SB-075 acetate SB-075 Diacetate SB-075 Cetrorelix Cetrorelix Diacetate Inhibitor SB-075 diacetate Gonadotropin releasing hormone receptor SB 075 Cetrorelix Acetate SB 075 Acetate Cetrorelix acetate SB-75 diacetate NS-75A diacetate SB075 inhibitor

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