Home Tools
Log in
Cart

Search Result

Search Results for " erβ "

20

Compounds

Cat No. Product Name Synonyms Targets
T2544 Bazedoxifene acetate WAY-TES 424,TSE 424,WAY-140424 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).
T6404 Bazedoxifene hydrochloride Bazedoxifene HCl,TSE-424 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bazedoxifene hydrochloride (TSE-424) is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectively.
T26537 AC-186 AC186,AC 186 Estrogen/progestogen Receptor
AC-186 is a nonsteroidal estrogen receptor β (ERβ) agonist with different affinities for ERβ and ERα, with an EC50 of 6 nM for ERβ and 5000 nM for ERα. AC-186 has neuroprotective activity and has been used in the study o...
T7644 DPN Diarylpropionitrile Apoptosis , Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Autophagy
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
T13443 (R)-Equol (+)-Equol Estrogen/progestogen Receptor
(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.
T3846 Bavachin Corylifolin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
T13674 Elacestrant RAD1901 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
T11915 LY88074 Estrogen/progestogen Receptor
LY88074 is a raloxifene analog in which the basic side chain has been removed. LY88074 is an agonist of ERβ (EC50 = 232 nM).This compound stimulates uterine cell proliferation.
T6533 Hexestrol Bibenzyl,Hexanoestrol,meso-Hexestrol,Hexestrofen Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Hexestrol (Hexanoestrol) binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
T23540 Y134 Y 134 Estrogen Receptor/ERR , Others
Y134 is an estrogen receptor inhibitor that is selective and orally active, exhibiting strong antagonist activity against ERα and Erβ with Ki of 0.09 nM and 11.31 nM, respectively. The selectivity of Y134 for ERα is 121...
T13675 Elacestrant dihydrochloride RAD1901 dihydrochloride Estrogen/progestogen Receptor
Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for ERβ, respectively.
T4000 (±)-Equol Equol,(R,S)-Equol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Drug Metabolite
(±)-Equol ((R,S)-Equol) is a non-steroidal estrogen produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. The estrogen receptor (ER) agonist activity of the naturally occu...
T4388 PHTPP Estrogen Receptor/ERR , Estrogen/progestogen Receptor
PHTPP is a selective ERβ antagonist.
T10239 Acolbifene EM-652,SCH 57068 Estrogen Receptor/ERR
Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifene shows an anticarcinogenic property.
T9800 Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- Estrogen/progestogen Receptor
Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.
T16566 Propyl pyrazole triol PPT Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: ...
T1048 Estradiol E2,17β-Estradiol,17β-Oestradiol,β-Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T3325 Liquiritigenin 4',7-Dihydroxyflavanone Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Liquiritigenin (4',7-Dihydroxyflavanone), a flavonoid aglycone from licorice, is a highly selective estrogen receptor β (ERβ) agonist.
T22794 G36 G-36 Estrogen Receptor/ERR
G36 is a cell-permeable non-steroidal antagonist of GPER. G36 inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 (IC50 = 112 and 165 nM, respectively). G36 has no detectable binding activity to...
T2250 DY131 DY 131,GSK 9089,DY-131 Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Smo
DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.

Compounds

Bazedoxifene acetate
T2544
Synonym: WAY-TES 424,TSE 424,WAY-140424
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Bazedoxifene hydrochloride
T6404
Synonym: Bazedoxifene HCl,TSE-424
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
AC-186
T26537
Synonym: AC186,AC 186
Target: Estrogen/progestogen Receptor
DPN
T7644
Synonym: Diarylpropionitrile
Target: Apoptosis, Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
(R)-Equol
T13443
Synonym: (+)-Equol
Target: Estrogen/progestogen Receptor
Bavachin
T3846
Synonym: Corylifolin
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Elacestrant
T13674
Synonym: RAD1901
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
LY88074
T11915
Synonym:
Target: Estrogen/progestogen Receptor
Hexestrol
T6533
Synonym: Bibenzyl,Hexanoestrol,meso-Hexestrol,Hexestrofen
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Y134
T23540
Synonym: Y 134
Target: Estrogen Receptor/ERR, Others
Elacestrant dihydrochloride
T13675
Synonym: RAD1901 dihydrochloride
Target: Estrogen/progestogen Receptor
(±)-Equol
T4000
Synonym: Equol,(R,S)-Equol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite
PHTPP
T4388
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Acolbifene
T10239
Synonym: EM-652,SCH 57068
Target: Estrogen Receptor/ERR
Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
T9800
Synonym:
Target: Estrogen/progestogen Receptor
Propyl pyrazole triol
T16566
Synonym: PPT
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Estradiol
T1048
Synonym: E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Liquiritigenin
T3325
Synonym: 4',7-Dihydroxyflavanone
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
G36
T22794
Synonym: G-36
Target: Estrogen Receptor/ERR
DY131
T2250
Synonym: DY 131,GSK 9089,DY-131
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Smo
1 2 3
TargetMol