20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9380 | Antide | ||
Antide has a wide range of applications in life science related research. | |||
T9380L | Antide acetate | Antide acetate (112568-12-4 Free base) | LHRH |
Antide acetate is an LHRH antagonist and represses LH and FSH release from the pituitary gland. | |||
TP1789L | Malantide acetate(86555-35-3 free base) | PKA , PKC | |
Malantide acetate is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activ... | |||
T15368L | Galantide acetate | Galantide acetate(138579-66-5 Free base) | Neuropeptide Y Receptor |
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two classes of galanin binding sites (KD<0.1 nM and ~6 nM) in t... | |||
TP2106L | Urantide acetate(669089-53-6 free base) | Neurotensin Receptor | |
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced ... | |||
T78556 | Antidepressant agent 5 | Others | |
Antidepressant agent 5 is a 7-substituted tetrahydroisoquinoline derivative with antidepressant activity.Antidepressant agent 5 acts similarly to magnoflorine in the study of depression and can be used for the prevention... | |||
T20413L | Spantide acetate | Spantide acetate(91224-37-2 Free base) | Neurokinin receptor |
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2. | |||
T75003 | Antidepressant agent 4 | ||
Antidepressant agent 4, an orally active compound, demonstrates efficacy as an antidepressant with additional anxiolytic, performance-enhancing, and nootropic activities [1]. | |||
TP2106 | Urantide | ||
Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acet... | |||
T75749 | Galantide TFA | ||
Galantide TFA, a reversible and non-specific antagonist of the galanin (GAL) receptor, demonstrates dose-dependent inhibition of galanin-induced K+ conductance, exhibiting an IC50 value of 4 nM. It is utilized in neurolo... | |||
T75002 | Antidepressant agent 3 | ||
Antidepressant agent 3, an orally active compound, showcases multifaceted pharmacological properties including antidepressant, anxiolytic, performance-enhancing, and nootropic activities [1]. | |||
TP2353 | Spantide II | ||
Spantide II is an antagonist of tachykinin. | |||
T19782 | Antidesmone | ||
Antidesmone is one compound mainly isolated from Ajugade cumbers Thunb (Labiatae). Antidesmone prevents acute lung injury via regulating MAPK and NF-κB activities. | |||
TP1789 | Malantide | ||
Malantide is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activity in v... | |||
T15368 | Galantide | Others | |
Galantide is a reversible and non-specific antagonist of galanin receptor. | |||
T62495 | Antidepressant agent 2 | ||
Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg. | |||
T82510 | Ecallantide TFA | DX-88 TFA | |
Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention of acute angioedema attacks [1]. | |||
T10332 | Antidepressant agent 1 | Others | |
Antidepressant agent 1 is a pyrazidole-halogeno-derivative with antidepressant effects. It also can be used to increase body temperature. | |||
T80031 | [D-Pro2] Spantide I TFA | Neurokinin receptor | |
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1]. | |||
T75837 | Spantide I TFA | ||
Spantide I TFA, a selective NK1 receptor antagonist and a substance P analog, exhibits K(i) values of 230 nM for NK1 and 8150 nM for NK2 receptors, respectively. It offers a method to decrease type 1 while increasing typ... |