keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 115.00 | |
5 mg | In stock | $ 233.00 | |
10 mg | In stock | $ 335.00 | |
25 mg | In stock | $ 565.00 | |
50 mg | In stock | $ 812.00 | |
100 mg | In stock | $ 1,130.00 |
Description | Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors). |
Molecular Weight | 1135.31 |
Formula | C53H70N10O14S2 |
CAS No. | TP2106L |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Urantide acetate(669089-53-6 free base) TP2106L GPCR/G Protein Neurotensin Receptor Urantide acetate(669089536 free base) Urantide acetate(669089 53 6 free base) inhibitor inhibit