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NH125

Catalog No. T6605    CAS 278603-08-0   

NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.

Pack Size Availability Price/USD Quantity
2 mg In stock 80.00
5 mg In stock 162.00
10 mg In stock 275.00
25 mg In stock 500.00
50 mg In stock 748.00
1 mL * 10 mM (in DMSO) In stock 296.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.

Receptor:

CaMKII; eEF-2 kinase; PKA; PKC;

Chemical Information:
Molecular Weight 524.56
Formula C27H45IN2
CAS Number 278603-08-0
Solubility

DMSO: 52.5 mg/mL (100 mM)

Ethanol: 39.3 mg/mL (75 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
Reference
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