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Cabergoline

Catalog No. T14853 CAS 81409-90-7

Synonyms: FCE-21336

Cabergoline is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively).Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Cabergoline, CAS 81409-90-7

Pack Size	Availability	Price/USD
2 mg	In stock	56.00
5 mg	In stock	81.00
10 mg	In stock	150.00
50 mg	In stock	449.00
100 mg	In stock	684.00
200 mg	In stock	1026.00

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Purity 99.92%

HNMR HPLC COA

Datasheet SDS

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Cabergoline is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively).Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.
Targets&IC50	Dopamine D2 receptor , Dopamine D3 receptor , 5-HT2B receptor

Synonyms	FCE-21336
Purity	99.92%
Molecular Weight	451.60
Formula	C26H37N5O2
CAS No.	81409-90-7

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 6 months

Solubility Information

DMSO: 32 mg/mL(70.86 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Odaka H, et al. Cabergoline, dopamine D2 receptor agonist, prevents neuronal cell death under oxidative stress via reducing excitotoxicity. PLoS One. 2014 Jun 10;9(6):e99271. 2. Jefferson F, et al. A dopamine receptor d2-type agonist attenuates the ability of stress to alter sleep in mice. Endocrinology. 2014 Nov;155(11):4411-21.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Clinical Compound Library Drug Repurposing Compound Library Neurotransmitter Receptor Compound Library Ferroptosis Compound Library

Related Products

Related compounds with same targets

Tandospirone GSK163090 Dexpramipexole Sumanirole maleate CP-809101 lumateperone Tosylate Nemifitide acetate(173240-15-8 free base) Neuromedin N acetate(92169-45-4 free base)

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.