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Search Results for " α2-adrenergic "

20

Compounds

Cat No. Product Name Synonyms Targets
T7045 Clonidine Nexiclon,Catapres,Kapvay Adrenergic Receptor
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-scale use for many years, clonidine has not been l...
T12643 (R)-Terazosin Adrenergic Receptor
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively).
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T6579 Medetomidine hydrochloride MPV785,Medetomidine HCl,Domitor Adrenergic Receptor
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
T0137 Mirtazapine 6-Azamianserin,Org3770 Dopamine Receptor , 5-HT Receptor , Opioid Receptor , Adrenergic Receptor , Histamine Receptor
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevations in serum aminotransferase levels and h...
T10052 AR-08 Adrenergic Receptor
AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.
T0505 Methyldopa L-(-)-α-Methyldopa,MK-351 Dopamine Receptor , Adrenergic Receptor
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
T4429 Rauwolscine hydrochloride Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride Adrenergic Receptor
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b...
T7065 Tizanidine Adrenergic Receptor
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.
T27599 Imiloxan RS-21361,RS 21361,RS21361 Adrenergic Receptor
Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.
T6766 Atipamezole Antisedan,MPV 1248 Adrenergic Receptor
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
T10100 QF0301B 5-HT Receptor , Adrenergic Receptor
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
T11894 Lusaperidone R107474 Adrenergic Receptor
Lusaperidone (R107474) is a potent α2-adrenergic receptor antagonist, a potential radioligand for the α (2)-adrenergic receptor, with inhibitory effects on α2A and α2C, with Ki values of 0.13 and 0.15 nM, respectively.
T23397 ST 91 Others , Adrenergic Receptor
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
T21371 Apraclonidine hydrochloride Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum Adrenergic Receptor
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pressure in human eyes and can be used in studies about glauco...
T16759 Ritanserin R 55667 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
T0290 Tizanidine hydrochloride Tizanidine HCl,DS 103-282 Adrenergic Receptor
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
T5954 Methyldopa hydrate Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate Dopamine Receptor , Adrenergic Receptor
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ...
T10998 Deriglidole SL 86-0715 Adrenergic Receptor
Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does not show activity against prazosin and rat co...
T34308 Rezatomidine AGN-203818,AGN203818,AGN 203818 Adrenergic Receptor
Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.

Compounds

Clonidine
T7045
Synonym: Nexiclon,Catapres,Kapvay
Target: Adrenergic Receptor
(R)-Terazosin
T12643
Synonym:
Target: Adrenergic Receptor
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Medetomidine hydrochloride
T6579
Synonym: MPV785,Medetomidine HCl,Domitor
Target: Adrenergic Receptor
Mirtazapine
T0137
Synonym: 6-Azamianserin,Org3770
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
AR-08
T10052
Synonym:
Target: Adrenergic Receptor
Methyldopa
T0505
Synonym: L-(-)-α-Methyldopa,MK-351
Target: Dopamine Receptor, Adrenergic Receptor
Rauwolscine hydrochloride
T4429
Synonym: Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
Tizanidine
T7065
Synonym:
Target: Adrenergic Receptor
Imiloxan
T27599
Synonym: RS-21361,RS 21361,RS21361
Target: Adrenergic Receptor
Atipamezole
T6766
Synonym: Antisedan,MPV 1248
Target: Adrenergic Receptor
QF0301B
T10100
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor
Lusaperidone
T11894
Synonym: R107474
Target: Adrenergic Receptor
ST 91
T23397
Synonym:
Target: Others, Adrenergic Receptor
Apraclonidine hydrochloride
T21371
Synonym: Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum
Target: Adrenergic Receptor
Ritanserin
T16759
Synonym: R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Tizanidine hydrochloride
T0290
Synonym: Tizanidine HCl,DS 103-282
Target: Adrenergic Receptor
Methyldopa hydrate
T5954
Synonym: Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate
Target: Dopamine Receptor, Adrenergic Receptor
Deriglidole
T10998
Synonym: SL 86-0715
Target: Adrenergic Receptor
Rezatomidine
T34308
Synonym: AGN-203818,AGN203818,AGN 203818
Target: Adrenergic Receptor
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TargetMol