20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7045 | Clonidine | Nexiclon,Catapres,Kapvay | Adrenergic Receptor |
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-scale use for many years, clonidine has not been l... | |||
T12643 | (R)-Terazosin | Adrenergic Receptor | |
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively). | |||
T3158 | Harmane | Loturine,Harman,Aribine | Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor |
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke. | |||
T6579 | Medetomidine hydrochloride | MPV785,Medetomidine HCl,Domitor | Adrenergic Receptor |
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor. | |||
T0137 | Mirtazapine | 6-Azamianserin,Org3770 | Dopamine Receptor , 5-HT Receptor , Opioid Receptor , Adrenergic Receptor , Histamine Receptor |
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevations in serum aminotransferase levels and h... | |||
T10052 | AR-08 | Adrenergic Receptor | |
AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit. | |||
T0505 | Methyldopa | L-(-)-α-Methyldopa,MK-351 | Dopamine Receptor , Adrenergic Receptor |
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic. | |||
T4429 | Rauwolscine hydrochloride | Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride | Adrenergic Receptor |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b... | |||
T7065 | Tizanidine | Adrenergic Receptor | |
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons. | |||
T27599 | Imiloxan | RS-21361,RS 21361,RS21361 | Adrenergic Receptor |
Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder. | |||
T6766 | Atipamezole | Antisedan,MPV 1248 | Adrenergic Receptor |
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. | |||
T10100 | QF0301B | 5-HT Receptor , Adrenergic Receptor | |
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors. | |||
T11894 | Lusaperidone | R107474 | Adrenergic Receptor |
Lusaperidone (R107474) is a potent α2-adrenergic receptor antagonist, a potential radioligand for the α (2)-adrenergic receptor, with inhibitory effects on α2A and α2C, with Ki values of 0.13 and 0.15 nM, respectively. | |||
T23397 | ST 91 | Others , Adrenergic Receptor | |
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile. | |||
T21371 | Apraclonidine hydrochloride | Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum | Adrenergic Receptor |
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pressure in human eyes and can be used in studies about glauco... | |||
T16759 | Ritanserin | R 55667 | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor |
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. | |||
T0290 | Tizanidine hydrochloride | Tizanidine HCl,DS 103-282 | Adrenergic Receptor |
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons. | |||
T5954 | Methyldopa hydrate | Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate | Dopamine Receptor , Adrenergic Receptor |
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ... | |||
T10998 | Deriglidole | SL 86-0715 | Adrenergic Receptor |
Deriglidole (SL 86-0715) is a peripheral adrenergic receptor antagonist that is a selective inhibitor of alpha2 receptors. Deriglidole inhibits colistin and Idazoxan but does not show activity against prazosin and rat co... | |||
T34308 | Rezatomidine | AGN-203818,AGN203818,AGN 203818 | Adrenergic Receptor |
Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain. |