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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN4442 | Linderene acetate | Prolyl Endopeptidase (PREP) | |
Linderene acetate is a competitive inhibitor against Prolyl endopeptidase. | |||
T2717 | Salidroside | Rhodioloside | Apoptosis , mTOR |
Salidroside (Rhodioloside) is a bioactive phenolic glycoside compound isolated from Rhodiola crenulata. It is a prolyl endopeptidase Inhibitor. | |||
T3891 | Oroxylin A-7-O-glucuronide | Oroxylin A Glucoronide,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide | Others |
Oroxylin A-7-O-glucuronide (Oroxylin A Glucoronide) and wogonoside should also be served as the chemical markers together with baicalin for the quality control of herbs and proprietary traditional Chinese medicine (PTCM)... | |||
T8657 | KYP-2047 | Others | |
KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor. | |||
T9855 | BR102910 | 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]- | Others |
BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) is a selective inhibitor of fibroblast activated protein (FAP). | |||
T2S0618 | β-Elemonic Acid | 3-oxo Tirucallic Acid,Beta-Elemonic acid,3-Oxotirucallenoic Acid,Elemadienonic Acid | Apoptosis , Reactive Oxygen Species , COX |
β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects. Beta-Elemonic acid inhibits proliferation by inducing hypoploid cells and cell apoptosis, the anticancer effects of beta-Elemonic acid are rel... | |||
T61622 | PREP inhibitor-1 | Others | |
PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease. | |||
T21011 | Buspirone | Buspirone free base,Ansial | 5-HT Receptor |
Buspirone (Buspirone free base) is an azaspiro compound which has a role as an anxiolytic drug, a sedative, a serotonergic agonist and an EC 3.4.21.26 (prolyl oligopeptidase) inhibitor. | |||
T7890 | SP-13786 | UAMC-1110 | Others |
SP-13786 (UAMC-1110) is an inhibitor of fibroblast activation protein (FAP) (IC50 : 3.2 nM); also inhibits prolyl oligopeptidase (PREP) ( IC50 : 1.8 μM). | |||
T78619 | Z-Pro-Pro-CHO | Prolyl Endopeptidase (PREP) | |
Z-Pro-Pro-CHO acts as a prolyl oligopeptidase inhibitor with half-maximal inhibitory concentrations (IC50) of 0.16 μM for human prolyl oligopeptidase and 0.01 μM for Schistosoma mansoni prolyl oligopeptidase [1]. | |||
TN3714 | (-)-Corypalmine | Corypalmine | Antifection |
Corypalmine (IC50=128.0±10.5 uM) can inhibit prolyl oligopeptidase. (-)-Corypalmine shows inhibition activity against spore germination of some fungi. | |||
T61995 | Y-29794 | ||
Y-29794 (Compound 2) is a potent, covalent inhibitor of prolyl oligopeptidase (POP) (Ki= 0.95 nM). Y-29794 has research value in neurodegenerative diseases and cancer. | |||
TN4426 | Leojaponin | AChR | |
Leojaponin is a prolyl oligopeptidase (POP) inhibitor. Leojaponin exhibits significant cytoprotective activities against glutamate-induced toxicity at concentrations ranging from 0.1 microm to 10 microm. | |||
T62534 | POP-IN-2 | ||
POP-IN-2 (Compound 7k) is a potent, covalently bound inhibitor of prolyl oligopeptidase (POP) (Ki: 6 nM).POP-IN-2 can be used in neurodegenerative disease and cancer research. | |||
T69603 | BR103354 | ||
BR103354 is a novel fibroblast activation protein (FAP) inhibitor with anti-diabetic and anti-steatotic effects. BR103354 inhibited FAP with an IC50 value of 14 nM, showing high selectivity against dipeptidyl peptidase (... |