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Search Results for " alpha-adrenergic "

20

Compounds

Cat No. Product Name Synonyms Targets
T2594 Dextromilnacipran Levomilnacipran Serotonin Transporter , Norepinephrine
Dextromilnacipran (Levomilnacipran) is a selective serotonin and norepinephrine reuptake inhibitor.
T5954 Methyldopa hydrate Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate Dopamine Receptor , Adrenergic Receptor
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ...
T0505 Methyldopa L-(-)-α-Methyldopa,MK-351 Dopamine Receptor , Adrenergic Receptor
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
T3046 BMY 7378 dihydrochloride BMY7378 HCl Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T4429 Rauwolscine hydrochloride Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride Adrenergic Receptor
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b...
T12030 MG 1 Adrenergic Receptor
MG 1 is a potent alpha-1 adrenergic receptor antagonist.
T8348 Phentolamine Adrenergic Receptor
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T3996 Dapiprazole Hydrochloride Glamidolo Hydrochloride,Reversil Hydrochloride Adrenergic Receptor
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, arterioles and veins), gastrointes...
T23283 2-Methoxyidazoxan monohydrochloride RX 821002 hydrochloride Adrenergic Receptor
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic effect on imidazoline. It has a significantly higher affinity ...
T5471 GUANABENZ Adrenergic Receptor
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T68023L Tolnapersine TFA Tolnapersine TFA(70312-00-4 Free base) Dopamine Receptor , Adrenergic Receptor
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
T1504 Silodosin KAD 3213,KMD 3213 Adrenergic Receptor
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
T1287 Synephrine Oxedrine Endogenous Metabolite , Adrenergic Receptor
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T1064 Norepinephrine bitartrate monohydrate Levophed,Noradrenaline bitartrate monohydrate Endogenous Metabolite , Adrenergic Receptor , Autophagy
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.
T1158 Phenoxybenzamine hydrochloride NCI-c01661,NSC 37448,Phenoxybenzamine HCl CaMK , Adrenergic Receptor
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and vasodilatory properties. Phenoxybenzamine non...
T0394 Moxisylyte hydrochloride Thymoxamine hydrochloride Adrenergic Receptor
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T21445 Naphazoline AK-Con,Naphcon-a,Clear Eyes,All Clear Adrenergic Receptor
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swelling when applied to mucous membrane.
T2150 Guanfacine hydrochloride Tenex,Intuniv,Guanfacine Adrenergic Receptor
Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
T22406 Prazosin Prazosine,Furazosin,Prazocin Adrenergic Receptor
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T22369 Midodrine (±)-Midodrin Adrenergic Receptor
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.

Compounds

Dextromilnacipran
T2594
Synonym: Levomilnacipran
Target: Serotonin Transporter, Norepinephrine
Methyldopa hydrate
T5954
Synonym: Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate
Target: Dopamine Receptor, Adrenergic Receptor
Methyldopa
T0505
Synonym: L-(-)-α-Methyldopa,MK-351
Target: Dopamine Receptor, Adrenergic Receptor
BMY 7378 dihydrochloride
T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Rauwolscine hydrochloride
T4429
Synonym: Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
MG 1
T12030
Synonym:
Target: Adrenergic Receptor
Phentolamine
T8348
Synonym:
Target: Adrenergic Receptor
Dapiprazole Hydrochloride
T3996
Synonym: Glamidolo Hydrochloride,Reversil Hydrochloride
Target: Adrenergic Receptor
2-Methoxyidazoxan monohydrochloride
T23283
Synonym: RX 821002 hydrochloride
Target: Adrenergic Receptor
GUANABENZ
T5471
Synonym:
Target: Adrenergic Receptor
Tolnapersine TFA
T68023L
Synonym: Tolnapersine TFA(70312-00-4 Free base)
Target: Dopamine Receptor, Adrenergic Receptor
Silodosin
T1504
Synonym: KAD 3213,KMD 3213
Target: Adrenergic Receptor
Synephrine
T1287
Synonym: Oxedrine
Target: Endogenous Metabolite, Adrenergic Receptor
Norepinephrine bitartrate monohydrate
T1064
Synonym: Levophed,Noradrenaline bitartrate monohydrate
Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy
Phenoxybenzamine hydrochloride
T1158
Synonym: NCI-c01661,NSC 37448,Phenoxybenzamine HCl
Target: CaMK, Adrenergic Receptor
Moxisylyte hydrochloride
T0394
Synonym: Thymoxamine hydrochloride
Target: Adrenergic Receptor
Naphazoline
T21445
Synonym: AK-Con,Naphcon-a,Clear Eyes,All Clear
Target: Adrenergic Receptor
Guanfacine hydrochloride
T2150
Synonym: Tenex,Intuniv,Guanfacine
Target: Adrenergic Receptor
Prazosin
T22406
Synonym: Prazosine,Furazosin,Prazocin
Target: Adrenergic Receptor
Midodrine
T22369
Synonym: (±)-Midodrin
Target: Adrenergic Receptor
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TargetMol