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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2594 | Dextromilnacipran | Levomilnacipran | Serotonin Transporter , Norepinephrine |
Dextromilnacipran (Levomilnacipran) is a selective serotonin and norepinephrine reuptake inhibitor. | |||
T5954 | Methyldopa hydrate | Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate | Dopamine Receptor , Adrenergic Receptor |
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ... | |||
T0505 | Methyldopa | L-(-)-α-Methyldopa,MK-351 | Dopamine Receptor , Adrenergic Receptor |
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic. | |||
T3046 | BMY 7378 dihydrochloride | BMY7378 HCl | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor |
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor. | |||
T4429 | Rauwolscine hydrochloride | Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride | Adrenergic Receptor |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b... | |||
T12030 | MG 1 | Adrenergic Receptor | |
MG 1 is a potent alpha-1 adrenergic receptor antagonist. | |||
T8348 | Phentolamine | Adrenergic Receptor | |
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist | |||
T3996 | Dapiprazole Hydrochloride | Glamidolo Hydrochloride,Reversil Hydrochloride | Adrenergic Receptor |
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, arterioles and veins), gastrointes... | |||
T23283 | 2-Methoxyidazoxan monohydrochloride | RX 821002 hydrochloride | Adrenergic Receptor |
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic effect on imidazoline. It has a significantly higher affinity ... | |||
T5471 | GUANABENZ | Adrenergic Receptor | |
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist. | |||
T68023L | Tolnapersine TFA | Tolnapersine TFA(70312-00-4 Free base) | Dopamine Receptor , Adrenergic Receptor |
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist. | |||
T1504 | Silodosin | KAD 3213,KMD 3213 | Adrenergic Receptor |
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist. | |||
T1287 | Synephrine | Oxedrine | Endogenous Metabolite , Adrenergic Receptor |
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma. | |||
T1064 | Norepinephrine bitartrate monohydrate | Levophed,Noradrenaline bitartrate monohydrate | Endogenous Metabolite , Adrenergic Receptor , Autophagy |
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator. | |||
T1158 | Phenoxybenzamine hydrochloride | NCI-c01661,NSC 37448,Phenoxybenzamine HCl | CaMK , Adrenergic Receptor |
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and vasodilatory properties. Phenoxybenzamine non... | |||
T0394 | Moxisylyte hydrochloride | Thymoxamine hydrochloride | Adrenergic Receptor |
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease. | |||
T21445 | Naphazoline | AK-Con,Naphcon-a,Clear Eyes,All Clear | Adrenergic Receptor |
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in reducing swelling when applied to mucous membrane. | |||
T2150 | Guanfacine hydrochloride | Tenex,Intuniv,Guanfacine | Adrenergic Receptor |
Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS. | |||
T22406 | Prazosin | Prazosine,Furazosin,Prazocin | Adrenergic Receptor |
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension. | |||
T22369 | Midodrine | (±)-Midodrin | Adrenergic Receptor |
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors. |