pca — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T13210	Trombodipine	PCA-4230	Antibiotic
	Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.		Antibiotic
T68644	Pca 4233
	Pca 4233 belongs to a class of selective PAF-receptor antagonists.
T33060	Lysine PCA
	Lysine PCA is a bioactive chemical.
T23123	PCA 4248		Others
	PAF antagonist		Others
T33356	Methylsilanol PCA
	Methylsilanol PCA is a bioactive chemical.
TP1037	D-Lys(Z)-Pro-Arg-pNA diacetate	Spectrozyme PCa,Chromozym Pca diacetate
	D-Lys(Z)-Pro-Arg-pNA (diacetate) diacetate is a chromogenic substrate.
TP1196	D-Lys(Z)-Pro-Arg-pNA	Chromozym Pca
	D-Lys(Z)-Pro-Arg-pNA is a luminescent substrate of activated protein C (APC).
T3160	HUHS015		Others
	HUHS015 is a potent PCA-1/ALKBH3 inhibitor.		Others
T13812	PCA50941		Others
	PCA50941 is a 1,4-dihydropyridine derivative, treatment for cardiovascular disease.		Others
T9593	Senaparib	IMP4297	PARP
	Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.		PARP
T3324	Lycorine	Galanthidine,Narcissine,Amarylline,Belamarine,Licorine	Apoptosis , Virus Protease , Antibacterial , AChR , Fatty Acid Synthase
	Lycorine (Narcissine) inhibits protein synthesis and may inhibit ascorbic acid biosynthesis, although studies on the latter are controversial and inconclusive.
T0860L	Mefloquine	Ro215998,WR 142490,Ro-215998,Lariam,Ro 215998	Others
	Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine is also a K+ channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine can be used for malaria, systemic l...		Others
T3049	TPCA-1	GW683965,IKK2 Inhibitor IV,TPCA1	Apoptosis , IκB/IKK , STAT
	TPCA-1 (TPCA1) is an effective and specific IKK-2 inhibitor (IC50: 17.9 nM); shows >22-fold selectivity over IKK-1 and >550-fold selectivity over others kinases and enzymes.		Apoptosis , IκB/IKK , STAT
T21653	1,4-DPCA		HIF/HIF Prolyl-Hydroxylase
	1,4-DPCA is an inhibitor of prolyl-hydroxylase with an IC50 of 2.4 µM for collagen hydroxylation in human foreskin fibroblasts and 60 μM for factor inhibiting HIF (FIH).		HIF/HIF Prolyl-Hydroxylase
T60452	PCAF-IN-2
	PCAF-IN-2 (compound 17) is a potent inhibitor of PCAF with an IC50 of 5.31 µM. PCAF-IN-2 exhibits anti-tumor activity. CAF-IN-2 induces cell apoptosis and arrest the cell cycle at the G2/M phase[1].
T60762	PCAF-IN-1
	PCAF-IN-1 is a antitumor agents used in tumor treatment research. PCAF-IN-1 is a highly selective inhibitor of PCAF [1].
T36796	1,4-DPCA ethyl ester
	1,4-DPCA ethyl ester, the ethyl ester derivative of 1,4-DPCA, acts as an inhibitor of the enzyme factor inhibiting HIF (FIH)[1].
T80282	CPcAMP1/26
	cPcAMP1/26, an antimicrobial peptide, exhibits potent bactericidal activity against A. hydrophila and S. aureus by inducing depolarization of the bacterial plasma membrane and elevating intracellular ROS (Reactive Oxygen...
T24146	HOCPCA
	HOCPCA is an effective and selective ligand for the GHB binding sites that acts by binding with 27 times better affinity than GHB itself and crossing the blood-brain barrier in vitro and in vivo.
T77552	SLU-PP-1072		Apoptosis , Estrogen/progestogen Receptor
	SLU-PP-1072 is an ERRα and ERRγ inverse dual agonist that disrupts PCa cell metabolism and induces apoptosis through cell cycle dysregulation.SLU-PP-1072 is used to study prostate cancer (PCa).		Apoptosis , Estrogen/progestogen Receptor