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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1146 | Nifedipine | BAY-a-1040,Procardia XL,Procardia,Adalat | CaMK , Potassium Channel , Calcium Channel , Autophagy |
Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent. Nifedipine inhibits the transmembrane influx of extracellular calcium ions into myocardial and vascular smooth muscle cells, causing dilatation ... | |||
T36665 | Dehydro Nifedipine | BAY-b 4759 | |
Dehydro Nifedipine (BAY-b 4759) is the main metabolite of nifedipine in human plasma. Dehydro Nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM. Nifedipine is a calcium channel blocker used i... | |||
T12222 | Nifedipine-d6 | Nifedipine D6,BAY-a-1040 D6 | Others |
Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel. | |||
T11926 | M-Nifedipine | Others | |
m-Nifedipine, an impurity of Nifedipine, serves as a potent calcium channel blocker and the preferred treatment option for cardiac insufficiencies. | |||
T69021 | Nifedipine HCl | ||
Nifedipine HCl is a potent vasodilator agent with calcium antagonistic action. It is a useful anti-anginal agent that also lowers blood pressure. | |||
T35584 | Hydroxydehydro Nifedipine Carboxylate | ||
Hydroxydehydro nifedipine carboxylate is a metabolite of nifedipine .1 1.Roosemalen, M.C.M., Soons, P.A., Funaki, T., et al.High-performance liquid chromatographic determination of the polar metabolites of nifedipine in ... | |||
T1215 | Nicardipine hydrochloride | RS-69216,Nicardipine HCl,YC-93 Hydrochloride | Calcium Channel , Adrenergic Receptor , AChR , Autophagy |
Nicardipine hydrochloride (YC-93 Hydrochloride) is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicardipine (Nifedipine Family) blocks cal... | |||
T0119 | Nitrendipine | BAY-E-5009,Bayotensin | Calcium Channel , Autophagy |
Nitrendipine (BAY-E-5009) is a calcium channel blocker with marked vasodilator action. It is an effective antihypertensive agent and differs from other calcium channel blockers in that it does not reduce glomerular filtr... | |||
T68972 | FR-7534 | ||
FR-7534 is a calcium antagonist structurally similar to nifedipine. | |||
T25010 | AK-2-38 | AK -2-38,AK2-38 | |
AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium. | |||
TN3147 | 6',7'-Dihydroxybergamottin | P450 | |
6',7'-Dihydroxybergamottin(DHB), a well-known inhibitor of CYP3A4, the inhibition of CYP3A4 activity by DHB includes the inhibition of POR activity, DHB can inhibit nifedipine oxidation in a concentration-dependent manne... | |||
TN3135 | 5-O-Methylnaringenin | Others | |
5-O-Methylnaringenin is a marker, reduced MS detection of 5-O-methylnaringenin indicated that nifedipine may preferably remove a proton from the 5-position OH group in the A ring of the flavonoid skeleton. | |||
T33673 | Niludipine | Niludipina,BAY-a 7168,Bay a 7168,Niludipinum | |
Nirudipine is a double (2-propoxyethyl) analogist of nifedipine and a calcium channel blocker, which is also a safe anti-angina Ca2+ antagonist with a broad range of efficacy for all types of angina. At the same time, Ni... | |||
T36070 | (±)5(6)-EET | ||
5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes. In solution, 5(6)-EET degrades into 5,6-DiHET and 5(6)-δ-lactone, which can be converted to 5... |