estrone — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T1009	Estrone	Oestrone,Fluoroethyl,Aquacrine	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Estrone (Aquacrine) is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone, a major mammalian estrogen. It is converted from ANDROSTENEDIONE directly, or from TESTOSTERONE via ESTRADIOL. In humans, it is pr...
T36857	Estrone sulfate sodium	Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate	Endogenous Metabolite
	Estrone sulfate sodium (17β-Estrone 3-sulfate) is an endogenous steroid and an estrogen ester that is biologically inactive. It is converted by steroid sulfatase into estrone . Estrone sulfate sodium has been investigate...		Endogenous Metabolite
T72470	Estrone O-sulfamate	Estrone 3-O-sulfamate	Others
	Estrone O-sulfamate (Estrone 3-O-sulfamate) is a potent inhibitor of steroid sulfatase (STS). Estrone O-sulfamate is a placental microsomal inhibitor (P.M.) with IC50 values of 18 nM. Estrone O-sulfamate showed inhibitor...		Others
T36857L	Premarin	Estrone 3-sulfate,Estrone sulfate	Estrogen Receptor/ERR
	Premarin (Estrone 3-sulfate) is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.		Estrogen Receptor/ERR
T0345	Estropipate	Piperazine estrone sulfate,Pipestrone,Estrone sulfate piperazine salt	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T73772	Estrone sulfate potassium		Endogenous Metabolite
	Estrone sulfate potassium is an estrogen ester and conjugate, a natural endogenous steroid.		Endogenous Metabolite
T36916	Estrone-3-Glucuronide (sodium salt hydrate)
	Estrone-3-Glucuronide is a metabolite of the primary premenopausal estrogen 17β-estradiol .1,2Urinary levels of estrone-3-Glucuronide peak approximately 36 hours prior to ovulation and have been used as a marker of ferti...
T28232	Oleoylestrone	Estrone 3-oleate,MP 101,MP-101,MP101	Antioxidant
	Oleoylestrone (MP-101) is present in plasma and adipose tissue, has potential antioxidant effects, induces loss of body fat in rats, and can be used for weight loss.		Antioxidant
T17940	Estrone-N-O-C1-amido	ERα ligand 1	Others
	Estrone-N-O-C1-amido (ERα ligand 1) is an estrogen ligand derived from Estrone that specifically binds to estrogen receptor α (ERα). Through a linker, Estrone-N-O-C1-amido (ERα ligand 1) forms a complex with the cIAP1 li...		Others
T73765	Estrone 3-glucuronide
	Estrone 3-glucuronide, a deuterium-labeled version, is recognized as the primary metabolite of estradiol and serves as a urinary marker for predicting the fertile window [1].
T9455	4-hydroxyestrone-4-methyl ether	4-Methoxy Estrone	Estrogen Receptor/ERR , Endogenous Metabolite
	4-hydroxyestrone-4-methyl ether (4-Methoxy Estrone) is the methylation of 4-OHE1, which is catalyzed by COMT.		Estrogen Receptor/ERR , Endogenous Metabolite
T9454	4-Hydroxyestrone		Estrogen Receptor/ERR , Endogenous Metabolite
	4-Hydroxyestrone, an endogenous estrogen metabolite, can strongly protect neuronal cells against oxidative damage.		Estrogen Receptor/ERR , Endogenous Metabolite
T13481	2-Methoxyestrone		Endogenous Metabolite
	2-Methoxyestrone is a methoxylated catechol estrogen and metabolite of estrone (pKa: 10.81).		Endogenous Metabolite
T36039	16α-Hydroxyestrone
	The naturally-occurring estrogens are estrone , estradiol , and estriol . 16α-hydroxy Estrone (16α-OHE1) is a hydroxylated metabolite of E1 as well as an interconversion product with E2. E1 is 16α-hydroxylated by cytochr...
T29886	Almestrone	BA-38372,BA 38372,Ciba-38372,BA38372,Ciba 38372
	Almestrone (developmental code names Ba 38372, Ciba 38372), also known as 7α-methylestrone, is a synthetic, steroidal estrogen which was synthesized in 1967 but was never marketed. It is used as a precursor in the synthe...
T11235	Estradiol 3-sulfamate	ES-J 995,E2MATE,BLE 00084	Others
	.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor.		Others
TQ0161	Mulberrin	Kuwanon C	Others
	Mulberrin (Kuwanon C) is an inhibitor of OATP2B1-mediated estrone-3-sulfate (E3S) uptake (IC50: 1.8 ±1.5 μM).		Others
T1571	Estriol	NSC-12169,Oestriol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , MRP , Endogenous Metabolite
	Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During PREGNANCY, a large amount of estriol is...
T36913	17-Epiestriol
	17-Epiestriol is a metabolite of estrone .1It is formed from estroneviaa 16α-hydroxy estrone intermediate by reduction of the C-17 ketone. 17-Epiestriol binds to estrogen receptor α (ERα) and ERβ with relative binding af...
T83766	Moexiprilat	RS 10029
	Moexiprilat, an active metabolite of the prodrug moexipril formed through side chain ester hydrolysis in vivo, functions as an angiotensin-converting enzyme (ACE; IC50 = 2.1 nM) inhibitor. At a concentration of 10 nM, it...