Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 78.00 | |
2 mg | In stock | $ 119.00 | |
5 mg | In stock | $ 178.00 | |
10 mg | In stock | $ 216.00 | |
25 mg | In stock | $ 475.00 | |
50 mg | In stock | $ 695.00 | |
100 mg | In stock | $ 988.00 | |
500 mg | In stock | $ 1,980.00 |
Description | Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor. |
In vivo | In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting[1]. |
Synonyms | Remoxipride Hydrochloride Anhydrous, Roxiam, (S)-Remoxipride Hydrochloride |
Molecular Weight | 407.73 |
Formula | C16H24BrClN2O3 |
CAS No. | 73220-03-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 40.9mg/mL (100mM)
You can also refer to dose conversion for different animals. More
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Remoxipride hydrochloride 73220-03-8 GPCR/G Protein Neuroscience Dopamine Receptor Remoxipride Hydrochloride Anhydrous Roxiam Remoxipride Hydrochloride (S)-Remoxipride Hydrochloride inhibitor inhibit