Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Phellopterin is a partial agonist of the central benzodiazepine receptors in vitro. Phellopterin shows a cytotoxic effect on RAW264.7 cell at the concentration from 40 to 400 μM. Phellopterin reduce TNF-alpha-induced VCAM-1 expression through regulation of the Akt and PKC pathway, which contributes to inhibit the adhesion of monocytes to endothelium.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 97.00 | |
5 mg | In stock | $ 163.00 | |
10 mg | In stock | $ 278.00 | |
25 mg | In stock | $ 475.00 | |
50 mg | In stock | $ 682.00 | |
100 mg | In stock | $ 948.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 178.00 |
Description | Phellopterin is a partial agonist of the central benzodiazepine receptors in vitro. Phellopterin shows a cytotoxic effect on RAW264.7 cell at the concentration from 40 to 400 μM. Phellopterin reduce TNF-alpha-induced VCAM-1 expression through regulation of the Akt and PKC pathway, which contributes to inhibit the adhesion of monocytes to endothelium. |
Source |
Molecular Weight | 300.31 |
Formula | C17H16O5 |
CAS No. | 2543-94-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (166.49 mM)
Chloroform: Soluble
You can also refer to dose conversion for different animals. More
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Phellopterin 2543-94-4 Membrane transporter/Ion channel Neuroscience GABA Receptor monocytes inhibit VCAM-1 endothelium Inhibitor inhibitor