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CP94253 hydrochloride

Catalog No. T22689 CAS 845861-39-4

Synonyms: CP 94253 hydrochloride

CP94253 hydrochloride (CP 94253 hydrochloride) is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

CP94253 hydrochloride Chemical Structure

CP94253 hydrochloride, CAS 845861-39-4

Pack Size	Availability	Price/USD
5 mg	In stock	$ 64.00
10 mg	In stock	$ 97.00
25 mg	In stock	$ 228.00
50 mg	In stock	$ 372.00
100 mg	In stock	$ 597.00
200 mg	In stock	$ 828.00
1 mL * 10 mM (in DMSO)	In stock	$ 64.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	CP 94253 hydrochloride
Molecular Weight	293.79
Formula	C15H20ClN3O
CAS No.	845861-39-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: < 7.34 mg/mL

DMSO: 120 mg/mL (408.46 mM), Sonication is recommended.

References and Literature

1. Knobelman DA, Kung HF, Lucki I. Regulation of extracellular concentrations of 5-hydroxytryptamine (5-HT) in mouse striatum by 5-HT(1A) and 5-HT(1B) receptors. J Pharmacol Exp Ther. 2000 Mar;292(3):1111-7 2. Koe et al (1992) Biochemical and behavioral studies of the 5-HT1B receptor agonist, CP-94,253. Drug Dev.Res. 26 241

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Membrane Protein-targeted Compound Library Neuronal Signaling Compound Library Bioactive Compound Library Neurotransmitter Receptor Compound Library Antidepressant Compound Library Anti-Cancer Compound Library Bioactive Compounds Library Max

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Related compounds with same targets

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

CP94253 hydrochloride 845861-39-4 GPCR/G Protein Neuroscience Others 5-HT Receptor CP94253 CP 94253 Hydrochloride CP-94253 Hydrochloride Serotonin Receptor inhibit CP 94253 CP-94253 CP 94253 hydrochloride 5-hydroxytryptamine Receptor Inhibitor CP94253 Hydrochloride inhibitor

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