δ-opioid — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T8991	BMS986187		Opioid Receptor
	BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.		Opioid Receptor
T4691	Asimadoline hydrochloride	EMD-61753 hydrochloride	Opioid Receptor
	Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also been shown to be used in the treatment of irritable bowel s...		Opioid Receptor
T4633	Asimadoline	EMD-61753	Opioid Receptor
	Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat peripheral pain such as arthritis. Asimadoline...		Opioid Receptor
TP1832	Gluten Exorphin C		Opioid Receptor
	Gluten exorphin C is an opioid peptide derived from wheat gluten. Its IC50 values are 40 μM and 13.5 μM for μ opioid and δ opioid activities in the GPI and MVD assays, respectively.Gluten Exorphin C, isolated from the pe...		Opioid Receptor
T7173L	[Leu5]-Enkephalin acetate(58822-25-6 free base)	Leucine enkephalin,Leu-enkephalin,Leucyl-enkephalin	Opioid Receptor , Endogenous Metabolite
	[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)		Opioid Receptor , Endogenous Metabolite
T7639	Deltorphin 2	Deltorphin 2(TFA),[D-Ala2]-Deltorphin II	Opioid Receptor
	Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.		Opioid Receptor
T6175	ADL-5859	ADL5859 Hydrochloride,ADL5859 HCl	Opioid Receptor
	ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the hERG channel.		Opioid Receptor
T4236	AR-M 1000390 hydrochloride	ARM390 Hydrochloride,ARM-390 HCl	Opioid Receptor
	AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic resp...		Opioid Receptor
T5167	Cebranopadol	GRT6005	Opioid Receptor
	Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP) and δ-opioid (DOP) receptor, respectively.		Opioid Receptor
T7637	Deltorphin I	Deltorphin 1,Deltorphin I(TFA),Deltorphin C	Opioid Receptor
	Deltorphin I is an agonist of δ-opioid receptor.		Opioid Receptor
TP1113L	[Leu5]-Enkephalin, amide acetate	[Leu5]-Enkephalin, amide acetate(60117-24-0 free base)	Opioid Receptor
	[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.		Opioid Receptor
T7173	[Leu5]-Enkephalin	Leucine enkephalin,Leucyl-enkephalin,Leu-enkephalin	Opioid Receptor , Endogenous Metabolite
	[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)		Opioid Receptor , Endogenous Metabolite
TP1254	[Met5]-Enkephalin, amide TFA	5-Methionine-enkephalin amide (TFA)	Opioid Receptor
	[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.		Opioid Receptor
TP1905	BW-180C	DADLE	Opioid Receptor
	BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.		Opioid Receptor
T23002	ML-335		Opioid Receptor
	ML-335 is a μ-δ isomer-targeted agonist, a μOR-δOR-biased ligand that can serve as a scaffold for the development of unique types of (isomer-biased) drugs.ML-335 is a MOR (μ-opioid receptor)/DOR (δ-opioid receptor) heter...		Opioid Receptor
T38193L	β-Endorphin (1-27) (human) acetate	β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)	Opioid Receptor
	β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity. β-Endorphin (1-27) (human) acetate is an agonist of opioid receptor, showing preferred affinity ...		Opioid Receptor
TP1367	[D-Ala2]leucine-enkephalin		Opioid Receptor
	[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.		Opioid Receptor
TP2105L	UFP-101 acetate	UFP-101 acetate(849024-68-6 free base)	Opioid Receptor
	UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.		Opioid Receptor
TP2036L	DPDPE TFA (88373-73-3 free base)	DPDPE TFA	Opioid Receptor
	DPDPE TFA is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinociceptive in vivo.		Opioid Receptor
T20435L	Leuphasyl TFA		Opioid Receptor
	Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors. Leuphasyl TFA is a potent, long-a...		Opioid Receptor