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Deltorphin 2

Catalog No. T7639 CAS 122752-16-3

Synonyms: Deltorphin 2(TFA), [D-Ala2]-Deltorphin II

Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Deltorphin 2, CAS 122752-16-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 57.00
5 mg	In stock	$ 177.00
10 mg	In stock	$ 327.00
25 mg	In stock	$ 555.00
50 mg	In stock	$ 798.00
100 mg	In stock	$ 1,090.00

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Purity: 100%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.
Targets&IC50	δ opioid receptor:0.41 nM

Synonyms	Deltorphin 2(TFA), [D-Ala2]-Deltorphin II
Molecular Weight	782.88
Formula	C38H54N8O10
CAS No.	122752-16-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 10mM

References and Literature

1. Thomas S A , Abbruscato T J , Hau V S , et al. Structure-Activity Relationships of a Series of [D-Ala2]Deltorphin I and II Analogues ;[J]. Journal of Pharmacology and Experimental Therapeutics, 1997, 281(2):817-825. 2. Willemse T, et al. Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings. Bioorg Med Chem Lett. 2018 Jul 15;28(13):2320-2323. doi: 10.1016/j.bmcl.2018.05.015. Epub 2018 May 12. Erratum in: Bioorg Med Chem Lett. 2018 Nov 1;28(20):3418.

Citations

1. Kan B F, Liu X Y, Han M M, et al.The NGF/TrKA pathway enhances analgesia in an experimental mice model of bone cancer pain by increasing membrane levels of δ-opioid receptors.Anesthesiology.2023:10-1097

Related compound libraries

This product is contained In the following compound libraries：

Anti-Neurodegenerative Disease Compound Library Peptide Compound Library Membrane Protein-targeted Compound Library GPCR Compound Library Endocrinology-Hormone Compound Library NO PAINS Compound Library Anti-Parkinson's Disease Compound Library Neuronal Signaling Compound Library Bioactive Compounds Library Max Bioactive Compound Library

Related Products

Related compounds with same targets

Naltrindole hydrochloride ORL1 antagonist 1 LY255582 CP-866087 JNJ-20788560 AR-M 1000390 hydrochloride Opioid receptor modulator 1 ADL-5859

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Keywords

Deltorphin 2 122752-16-3 Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor Deltorphin 2(TFA) inhibit Deltorphin2 Inhibitor [D-Ala2]-Deltorphin II Deltorphin-2 inhibitor

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