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Search Results for " parasympathomimetic "

15

Compounds

Cat No. Product Name Synonyms Targets
T2390 Cevimeline hydrochloride hemihydrate AChR
Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.
T0229 Rivastigmine SDZ-ENA 713,S-Rivastigmine,Exelon AChE
Rivastigmine (Exelon) is a Cholinesterase Inhibitor, used for therapy of Alzheimer disease.
T3126 Bethanechol chloride (±)-Bethanechol,Urecholine,Myocholine,Carbamyl-β-methylcholine chloride AChR
Bethanechol chloride (Carbamyl-β-methylcholine chloride) is a slowly hydrolyzing muscarinic agonist with no nicotinic effects. Bethanechol is generally used to increase smooth muscle tone, as in the GI tract following ab...
T1628 Rivastigmine tartrate SDZ-ENA 713,ENA 713 AChR , AChE
Rivastigmine tartrate (SDZ-ENA 713) is a carbamate-derived reversible CHOLINESTERASE INHIBITOR that is selective for the CENTRAL NERVOUS SYSTEM and is used for the treatment of DEMENTIA in ALZHEIMER DISEASE and PARKINSON...
T0130 Physostigmine Salicylate AChR , AChE
Physostigmine, a parasympathomimetic alkaloid, is a reversible cholinesterase inhibitor. It extracts from the Calabar bean.
T1682 Methacholine Chloride Mecholyl chloride,Acetyl-β-methylcholine chloride AChR
Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of ACETYLCHOLINE. It is hydrolyzed by ACETYLCHOLINESTERASE at a considerably slower r...
T1221 Acetylcholine chloride ACh chloride,Pilofrin Calcium Channel , Endogenous Metabolite , AChR
Acetylcholine Chloride is the chloride salt form of acetylcholine, a synthetic, quaternary amino alcohol with cholinergic properties. Acetylcholine chloride (Pilofrin) mimics the parasympathomimetic effect of the endogen...
T4439 Sn-Glycero-3-phosphocholine Choline Alfoscerate,Glycerophosphocholine,Glycerophosphorylcholine,Alpha-GPC,Choline glycerophosphate,L-α-GPC Endogenous Metabolite , AChE
sn-Glycero-3-phosphocholine (Choline glycerophosphate) is a natural choline compound found in the brain and in milk. It is also a parasympathomimetic acetylcholine precursor which may have a potential for the treatment o...
T22296 Cisapride hydrate Propulsid,Alimix,Enteropride,Kinestase,Propulsin EGFR , 5-HT Receptor
Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.
T12587 Pyridostigmine-d6 bromide Pyridostigmine D6 bromide Others
Pyridostigmine D6 bromide is the deuterium labeled Pyridostigmine, which is a parasympathomimetic and a reversible inhibitor of cholinesterase.
T70311 Demecarium Free Base
Demecarium Free Base is a quaternary ammonium compound that serves as a long-acting cholinesterase inhibitor with parasympathomimetic activity. When used topically, demecarium inactivates both pseudocholinesterase and ac...
T21119 Cevimeline AF-102B,FKS 508,SNI 2011,HSDB 7286
Cevimeline, a parasympathomimetic and muscarinic agonist, affects M1 and M3 receptors. Cevimeline has been shown to treat dry mouth and Sj gren's syndrome. It is also used to reduce Xerostomia symptoms and increase saliv...
T68116 Norcisapride
Norcisapride belongs to the class of organic compounds known as diphenylpyrroles. Norcisapride acts directly as a serotonin 5-HT4 receptor agonist and indirectly as a parasympathomimetic. Norcisapride is a metabolite of ...
T69158 Ambenonium chloride tetrahydrate
Ambenonium chloride tetrahydrate is a salt of ambenonium --- a quaternary ammonium compound with parasympathomimetic activity. It is a cholinesterase inhibitor used in the management of myasthenia gravis. Myasthenia grav...
T71758 Ambenonium chloride
Ambenonium Chloride is the chloride salt form of ambenonium, a quaternary ammonium compound with parasympathomimetic activity. It is a cholinesterase inhibitor used in the management of myasthenia gravis. Myasthenia grav...
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