taar1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T9357	Ro 5212773	Epptb	Others
	Ro 5212773 (Epptb) is a selective TAAR1 antagonist.		Others
T9183	Ralmitaront	RO6889450	Others
	Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).		Others
T34374	RO5203648 HCl	RO5203648,RO-5203648,RO 5203648	Others
	RO5203648 HCl is a partial agonist of trace amine-related receptor 1 (TAAR1) with antipsychotic and antidepressant-like activities. RO5203648 HCl can be used in studies about neuropsychiatric therapeutics.		Others
T34373	RO5166017	RO 5166017,RO-5166017	Others
	RO5166017 is an orally active, potent and selective trace amine-associated receptor 1 (TAAR1) agonist for the study of conditioned taste aversion frontal nerve disorders.		Others
T12745	RO5263397		Others
	RO5263397 is a TAAR1 specific agonist with oral activity that has been used in antidepressant studies. It has also been found to act as an inhibitor of the enzyme cyclooxygenase-2 (COX-2), which is involved in the synthe...		Others
T4710	3-Methoxytyramine hydrochloride	3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride)	Others , Endogenous Metabolite , Drug Metabolite
	3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) is an inactive metabolite of dopamine which can activate trace amine associated receptor 1 (TAAR1). 3-methoxytyramine can be found primarily in human br...		Others , Endogenous Metabolite , Drug Metabolite
T0647	Tryptamine		Dehydrogenase , 5-HT Receptor , Endogenous Metabolite , TRP/TRPV Channel
	Tryptamine is a monoamine alkaloid found in animals, plants, and fungi. It contains an indole ring structure and is structurally analogous to the tryptophan. It is found in trace amounts in the brains of mammals and is r...
T3095	Tyramine	4-hydroxyphenethylamine,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine	MAO , Endogenous Metabolite
	Tyramine (Uteramine) is an indirect sympathomimetic that occurs naturally in cheese and other foods. Tyramine does not directly activate adrenergic receptors, but it can serve as a substrate for adrenergic uptake systems...		MAO , Endogenous Metabolite
T71606	RO5073012
	RO5073012 is a novel potent and selective TAAR1 partial agonist.
T80733	ZH8667
	ZH8667 is a TAAR1-Gs agonist that holds potential for schizophrenia research [1].
T12744	RO5256390		Others
	RO5256390 is a trace amine-associated receptor 1 (TAAR1) agonist, a highly conserved G-protein-coupled receptor that blocks psychostimulant-induced hyperarousal, and may be used in the study of neurological disorders.		Others
T80734	ZH8659
	ZH8659 is a Gq agonist targeting the trace amine-associated receptor 1 (TAAR1) and has potential applications in schizophrenia research [1].
T38172	RO 5263397 hydrochloride
	Potent trace amine 1 (TA1) receptor agonist (EC50 values are 0.12, 35 and 17-85 nM for mouse, rat and human receptors, respectively). Increases wakefulness and reduces REM and NREM sleep duration in wild type mice. Inhib...
T12899L	SEP-363856 hydrochloride	SEP-856 hydrochloride	Others , 5-HT Receptor
	SEP-363856 hydrochloride (SEP-856 hydrochloride) is an agent of orally active and CNS active psychotropic with a unique, non-D2/5-HT2A mechanism of action, exerts its antipsychotic-like effects, has the potential to trea...		Others , 5-HT Receptor
T12899	SEP-363856	SEP-856	Others
	SEP-363856 is an agent of orally active and CNS active psychotropic with a unique, non-D2/5-HT2A mechanism of action, exerts its antipsychotic-like effects, has the potential to treatment of schizophrenia.		Others