Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ro 5212773 (Epptb) is a selective TAAR1 antagonist.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 31.00 | |
5 mg | In stock | $ 72.00 | |
10 mg | In stock | $ 128.00 | |
25 mg | In stock | $ 285.00 | |
50 mg | In stock | $ 570.00 | |
100 mg | In stock | $ 817.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 79.00 |
Description | Ro 5212773 (Epptb) is a selective TAAR1 antagonist. |
Targets&IC50 | TAAR1:28 nM |
In vivo | EPPTB prevents the reduction of the firing frequency of DA neurons induced by p-tyramine (p-tyr), a nonselective TAAR1 agonist. the EPPTB effects were absent in Taar1 knockout mice, ruling out off-target effects[2]. |
Synonyms | Epptb |
Molecular Weight | 378.39 |
Formula | C20H21F3N2O2 |
CAS No. | 1110781-88-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/ml (145.35 mM)
You can also refer to dose conversion for different animals. More
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Ro 5212773 1110781-88-8 Others Ro-5212773 Inhibitor Epptb neuronal inhibit Ro5212773 mesolimbic system TAAR1 GPCR inhibitor