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20

Compounds

Cat No. Product Name Synonyms Targets
T10379 Arzoxifene hydrochloride SERM 3,LY 353381 HCl Others
Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.
T2544 Bazedoxifene acetate WAY-TES 424,TSE 424,WAY-140424 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).
T6404 Bazedoxifene hydrochloride Bazedoxifene HCl,TSE-424 Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Bazedoxifene hydrochloride (TSE-424) is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectively.
T73702 Mecasermin
Mecasermin (Human IGF-I; FK 780), a recombinant form of human insulin-like growth factor I (IGF-I), holds promise for investigating growth failure attributed to growth hormone (GH) insensitivity, which may be due to defe...
T24002 Disermolide XAA 296,XAA296,XAA-296
Disermolide is a polyketide natural product found to stabilize microtubules. Disermolide was found to be a potent inhibitor of tumor cell growth in several MDR cancer cell lines.
T26186 Sermetacin Sermetacina,SH G 318 AB,SHG 318 AB,TVX 3158
Sermetacin is an anti-inflammatory agent.
T25534 Indazole-Cl Indazole Cl Estrogen/progestogen Receptor
Indazole-Cl is a selective ERß agonist and a selective estrogen receptor modifier (SERM).
T27322 Fispemifene HM-101,HM 101,HM101 Others
Fispemifene (HM-101) is an estrogen receptor modulator (SERM) used to treat genitourinary syndromes and vaginal atrophy.
T4420 4-Hydroxytamoxifen ICI 79280,(Z)-4-hydroxy Tamoxifen,trans-4-Hydroxytamoxifen Estrogen Receptor/ERR , Estrogen/progestogen Receptor
4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency. 4-Hydroxytamoxifen has antitumor activity and may be used in breast cancer rese...
T15249 Estrogen receptor modulator 1 Estrogen Receptor/ERR
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.4...
T1549 Raloxifene hydrochloride LY156758 hydrochloride,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl Estrogen Receptor/ERR , Others , MAO , Estrogen/progestogen Receptor , Autophagy
Raloxifene hydrochloride (LY156758 hydrochloride) is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estrogen agonist effects on bone and chol...
T2569 Chlorotrianisene tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE Estrogen Receptor/ERR , Estrogen/progestogen Receptor , COX
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but...
T6620 Ospemifene FC-1271a Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Ospemifene (FC-1271a) is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA ap...
T7839 Lasofoxifene Tartrate CP-336156 Estrogen Receptor/ERR
Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.
T28957 TFR4OHT TFR-4-OHT,TFR 4 OHT
TFR4OHT is a selective ER modulator (SERM).
T25700L Levormeloxifene fumarate
Levormeloxifene fumarate is an osteoporosis drug and selective estrogen receptor modulator (SERM).
T3645 Endoxifen E-isomer hydrochloride E-Endoxifen hydrochloride Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
T27946 LY-329146 LY 329146
LY-329146 is a selective estrogen receptor modulator (SERM). LY-329146 prevents doxorubicin resistance in tumor cells expressing multidrug resistance-associated protein (MRP) by inhibiting the binding of MRP substrates t...
T13076 Tamoxifen-​d5 ICI 47699-​d5,(Z)-Tamoxifen-​d5,trans-Tamoxifen-​d5 HSP
Tamoxifen-d5 is a deuterium labeled Tamoxifen. Tamoxifen is a selective modulator of estrogen receptor (SERM). Tamoxifen is a potent activator of Hsp90 and enhances the Hsp90 molecular chaperone ATPase activity.
T62119 Lasofoxifene
Lasofoxifene (CP-336156) is a selective, orally active estrogen receptor modulator (SERM) that inhibits the growth and metastasis of primary tumours and is also anti-osteoporotic.

Compounds

Arzoxifene hydrochloride
T10379
Synonym: SERM 3,LY 353381 HCl
Target: Others
Bazedoxifene acetate
T2544
Synonym: WAY-TES 424,TSE 424,WAY-140424
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Bazedoxifene hydrochloride
T6404
Synonym: Bazedoxifene HCl,TSE-424
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Mecasermin
T73702
Synonym:
Target:
Disermolide
T24002
Synonym: XAA 296,XAA296,XAA-296
Target:
Sermetacin
T26186
Synonym: Sermetacina,SH G 318 AB,SHG 318 AB,TVX 3158
Target:
Indazole-Cl
T25534
Synonym: Indazole Cl
Target: Estrogen/progestogen Receptor
Fispemifene
T27322
Synonym: HM-101,HM 101,HM101
Target: Others
4-Hydroxytamoxifen
T4420
Synonym: ICI 79280,(Z)-4-hydroxy Tamoxifen,trans-4-Hydroxytamoxifen
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Estrogen receptor modulator 1
T15249
Synonym:
Target: Estrogen Receptor/ERR
Raloxifene hydrochloride
T1549
Synonym: LY156758 hydrochloride,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Chlorotrianisene
T2569
Synonym: tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, COX
Ospemifene
T6620
Synonym: FC-1271a
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Lasofoxifene Tartrate
T7839
Synonym: CP-336156
Target: Estrogen Receptor/ERR
TFR4OHT
T28957
Synonym: TFR-4-OHT,TFR 4 OHT
Target:
Levormeloxifene fumarate
T25700L
Synonym:
Target:
Endoxifen E-isomer hydrochloride
T3645
Synonym: E-Endoxifen hydrochloride
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
LY-329146
T27946
Synonym: LY 329146
Target:
Tamoxifen-​d5
T13076
Synonym: ICI 47699-​d5,(Z)-Tamoxifen-​d5,trans-Tamoxifen-​d5
Target: HSP
Lasofoxifene
T62119
Synonym:
Target:
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TargetMol