12
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T23490 | UBP310 | UBP 310 | Others , iGluR |
UBP310 (UBP 310) is a GLUK5 kainate receptor antagonist | |||
T81801 | MGluR5 antagonist-1 | ||
mGluR5 antagonist-1 (compound 10) is a potent mGluR5 inhibitor exhibiting an IC50 of 11.5 nM and demonstrates antidepressant effects [1]. | |||
T38659 | MGluR5 modulator 1 | ||
mGluR5 modulator 1 is a compound that acts as a positive allosteric modulator of the metabotropic glutamate receptor subtype 5 (mGluR5). Its primary application lies in the field of schizophrenia and cognitive impairment... | |||
T27947L | LY339434 HCl | LY339434 HCl(219566-62-8 Free base) | GluR , NMDAR |
LY339434 HCl is a low affinity GluR5 erythrocyte receptor agonist.LY339434 HCl causes rapid neuronal death primarily by affecting N-methyl-D-aspartate (NMDA) receptors. | |||
T27949 | LY382884 | LY-382884,LY 382884 | GluR |
LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction. | |||
T0675 | Topiramate | RWJ 17021,McN 4853 | Potassium Channel , Calcium Channel , GABA Receptor , Sodium Channel , GluR , Carbonic Anhydrase , iGluR |
Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures. Topiramate has been rarely associated with hepatic injury and largely when used in combination ... | |||
T10405 | ATPA | Others | |
ATPA is a selective glutamate receptor GluR5 activator (EC50s: 0.66, 1.4, 9.5, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S721T), GluR5(S741M), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V)). | |||
T27947 | LY339434 | LY 339434,LY-339434 | |
LY339434 is a potent and selective agonist of the kainate receptor GluK1, GluR5. | |||
T23488 | UBP 296 | Others | |
GluR5-subunit containing kainate receptor antagonist | |||
T22546 | UBP316 | ACET | Others |
GluR5-containing kainate receptor antagonist | |||
T13185 | Topiramate D12 | RWJ 17021 D12,McN 4853 D12 | Others |
Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor. | |||
T61145 | Topiramate lithium | ||
Topiramate lithium (McN 4853) is a wide-ranging antiepileptic compound with GluR5 receptor antagonistic properties. Its mechanism of action involves enhancing GABAergic activity, inhibiting kainate/AMPA receptors, voltag... |