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Nociceptin (1-13), amide

Catalog No. TP1793 CAS 178064-02-3

Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.

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Nociceptin (1-13), amide Chemical Structure

Nociceptin (1-13), amide, CAS 178064-02-3

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10 mg	Inquiry	$ 152.00
25 mg	Inquiry	$ 229.00
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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes.

Molecular Weight	1381.59
Formula	C61H100N22O15
CAS No.	178064-02-3

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Varani K, et al. Nociceptin receptor binding in mouse forebrain membranes: thermodynamic characteristics and structure activity relationships. Br J Pharmacol. 1998 Dec;125(7):1485-90.

Related Products

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Sideritoflavone PZM21 Nociceptin (1-13) amide TFA Ac-RYYRIK-NH2 acetate Ac-RYYRWK-NH2 acetate Naltrexone hydrochloride Samidorphan HCl Opioid receptor modulator 1

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Keywords

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