Powder: -20°C for 3 years | In solvent: -80°C for 1 year
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 38.00 | |
2 mg | In stock | $ 54.00 | |
5 mg | In stock | $ 88.00 | |
10 mg | In stock | $ 129.00 | |
25 mg | In stock | $ 247.00 | |
50 mg | In stock | $ 398.00 | |
100 mg | In stock | $ 592.00 | |
500 mg | In stock | $ 1,280.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 97.00 |
Description | JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM. |
Targets&IC50 | α2C-adrenoceptor: 28 nM (ki), α2C-adrenoceptor:16 nM (kb) |
Molecular Weight | 441.4 |
Formula | C24H26Cl2N4 |
CAS No. | 1259314-65-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 12 mg/mL (27.18 mM), Sonication is recommended.
DMSO: 5 mg/mL (11.33 mM), when pH is adjusted to 5 with NaOH. Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
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