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GR 125743

GR 125743
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
Catalog No. T8737Cas No. 148547-33-5
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Purity:99.76%
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GR 125743

Catalog No. T8737Cas No. 148547-33-5
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
1 mg$36In Stock
2 mg$51In Stock
5 mg$80In Stock
10 mg$122In Stock
25 mg$247In Stock
50 mg$369In Stock
100 mg$549In Stock
1 mL x 10 mM (in DMSO)$89In Stock
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Product Introduction

Bioactivity
Description
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
In vitro
GR-125743, a new radiolabelled derivative of a compound that exhibits selective antagonistic properties with respect to the serotonin human (h5-HT1D) and human (h5-HT1B) receptors.?The compound has been characterized for its ability to label the cloned h5-HT1D and h5-HT1B receptors.
Chemical Properties
Molecular Weight416.52
FormulaC25H28N4O2
Cas No.148547-33-5
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 4.17 mg/mL (10 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4008 mL12.0042 mL24.0085 mL120.0423 mL
5 mM0.4802 mL2.4008 mL4.8017 mL24.0085 mL
10 mM0.2401 mL1.2004 mL2.4008 mL12.0042 mL

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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