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Search Results for " α1-adrenoceptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T10003 α1 adrenoceptor-MO-1 Others
α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.
T12643 (R)-Terazosin Adrenergic Receptor
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values of 6.51 nM, 1.01 nM and 1.97 nM, respectively).
T0197 Terazosin hydrochloride Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic Adrenergic Receptor
Terazosin hydrochloride (Hytrin) , a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for patients with prostate enlargement and h...
T6701 Terazosin hydrochloride dihydrate Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate Adrenergic Receptor
Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
T0088 Urapidil hydrochloride Urapidil HCl 5-HT Receptor , Adrenergic Receptor
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T12597 5-HT2 antagonist 1 5-HT Receptor
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
T61535 Neldazosin Adrenergic Receptor
Neldazosin is used as a potent α1-adrenoceptor antagonist.
T28922 Taprizosin Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003 Adrenergic Receptor
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.
T6600 Naftopidil dihydrochloride KT-611,KT-611 2HCl,Naftopidil DiHCl 5-HT Receptor , Adrenergic Receptor
Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T17310 Phenylephrine L-Phenylephrine,(R)-(-)-Phenylephrine Adrenergic Receptor
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T6579 Medetomidine hydrochloride MPV785,Medetomidine HCl,Domitor Adrenergic Receptor
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
T11015 Midaglizole hydrochloride (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128 Adrenergic Receptor
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenocepto...
T0165 Urapidil Mediatensyl,Ebrantil,Eupressyl 5-HT Receptor , Adrenergic Receptor
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T11286 Fiduxosin A 185980.1,ABT 980 Adrenergic Receptor
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin...
T23232 Remoxipride hydrochloride Remoxipride Hydrochloride Anhydrous,Roxiam,(S)-Remoxipride Hydrochloride Dopamine Receptor
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
T9762 Upidosin SB-216469,SB 216469,Rec 15-2739,Recordati 15/2739 Adrenergic Receptor
Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM.
T62893 SM-2470 Adrenergic Receptor
SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity that decreases anterior ganglionic adrenal nerve activity and aortic descending nerve activity.SM-2470 has hypocholesterolemic activity and inhibits...
T8044 Ajmalicine Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin Adrenergic Receptor
Ajmalicine (Raubasine) (Raubasine) is a potent adrenolytic agent which preferentially blocks α1-adrenoceptor. Ajmalicine is an reversible but non-competitive nicotine receptor full inhibitor, IC50 = 72.3 μM. Ajmalicine a...
T0696 Naftopidil KT-611,BM-15275 Adrenergic Receptor
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
T9220 Naftopidil hydrochloride 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride Adrenergic Receptor
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, respective...

Compounds

α1 adrenoceptor-MO-1
T10003
Synonym:
Target: Others
(R)-Terazosin
T12643
Synonym:
Target: Adrenergic Receptor
Terazosin hydrochloride
T0197
Synonym: Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic
Target: Adrenergic Receptor
Terazosin hydrochloride dihydrate
T6701
Synonym: Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate
Target: Adrenergic Receptor
Urapidil hydrochloride
T0088
Synonym: Urapidil HCl
Target: 5-HT Receptor, Adrenergic Receptor
5-HT2 antagonist 1
T12597
Synonym:
Target: 5-HT Receptor
Neldazosin
T61535
Synonym:
Target: Adrenergic Receptor
Taprizosin
T28922
Synonym: Taprizosin Mesylate,UK-338003,UK-338,003,UK338003,UK 338003
Target: Adrenergic Receptor
Naftopidil dihydrochloride
T6600
Synonym: KT-611,KT-611 2HCl,Naftopidil DiHCl
Target: 5-HT Receptor, Adrenergic Receptor
Phenylephrine
T17310
Synonym: L-Phenylephrine,(R)-(-)-Phenylephrine
Target: Adrenergic Receptor
Medetomidine hydrochloride
T6579
Synonym: MPV785,Medetomidine HCl,Domitor
Target: Adrenergic Receptor
Midaglizole hydrochloride
T11015
Synonym: (±)-DG5128,(±)-DG5128 hydrochloride,DG5128 hydrochloride,DG5128
Target: Adrenergic Receptor
Urapidil
T0165
Synonym: Mediatensyl,Ebrantil,Eupressyl
Target: 5-HT Receptor, Adrenergic Receptor
Fiduxosin
T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Remoxipride hydrochloride
T23232
Synonym: Remoxipride Hydrochloride Anhydrous,Roxiam,(S)-Remoxipride Hydrochloride
Target: Dopamine Receptor
Upidosin
T9762
Synonym: SB-216469,SB 216469,Rec 15-2739,Recordati 15/2739
Target: Adrenergic Receptor
SM-2470
T62893
Synonym:
Target: Adrenergic Receptor
Ajmalicine
T8044
Synonym: Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin
Target: Adrenergic Receptor
Naftopidil
T0696
Synonym: KT-611,BM-15275
Target: Adrenergic Receptor
Naftopidil hydrochloride
T9220
Synonym: 1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,KT-611 hydrochloride,BM-15275 hydrochloride
Target: Adrenergic Receptor
1 2 3
TargetMol