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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1069 | Metoclopramide hydrochloride | Maxolon,Metoclopramide HCl | Dopamine Receptor , 5-HT Receptor , AChR |
Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic. | |||
T4616 | Metoclopramide | 5-Chloro-2-methoxyprocainamide | Dopamine Receptor , 5-HT Receptor |
Metoclopramide (5-Chloro-2-methoxyprocainamide) is a dopamine D2 antagonist which has been used for treatment of a variety of gastrointestinal symptoms over the last thirty years. In various countries, metoclopramide is ... | |||
T8385 | Metoclopramide hydrochloride hydrate | Metoclopramide monohydrochloride monohydrate | Dopamine Receptor , 5-HT Receptor |
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It acts as an anti-emetic | |||
T1528 | Azasetron hydrochloride | Y-25130 hydrochloride,Y-25130 HCl,Azasetron HCl | 5-HT Receptor |
Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic. | |||
T11326 | Frovatriptan succinate hydrate | Frovelan,Frova | 5-HT Receptor |
Frovatriptan succinate hydrate (Frova) is effective in treating the full spectrum of migraine including the associated symptoms of nausea, vomiting, photophobia, and phonophobia. Frovatriptan succinate hydrate can also b... | |||
T1478 | Ondansetron hydrochloride dihydrate | SN 307,NSC 665799,GR 38032,Ondansetron hydrochloride | 5-HT Receptor |
Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, a... | |||
T1790 | Fosaprepitant dimeglumine | L785298,MK-0517,Fosaprepitant dimeglumine salt | Neurokinin receptor |
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic activity. Upon intravenous administration and rapid conversion... | |||
T16433 | Pancopride | LAS 30451 | 5-HT Receptor |
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced vomiting. | |||
T13329L | Vofopitant dihydrochloride | GR 205171A,Vofopitant 2HCl | Neurokinin receptor |
Vofopitant dihydrochloride (GR 205171A) is an orally available, selective tachykinin NK1 receptor antagonist that inhibits [3H]SP binding to NK1 with pKi values of 9.5 and 10.6, respectively.Vofopitant dihydrochloride is... | |||
T28187 | Nonabine | ||
Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy. | |||
T22313 | Dolasetron Mesylate | Anzemet hydrate,MDL-73147EF | Others , 5-HT Receptor |
Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following chemotherapy. | |||
T7569 | Clebopride malate | Dopamine Receptor | |
Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting. | |||
T2574 | Alizapride hydrochloride | Alizapride HCl | Dopamine Receptor |
Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting. | |||
T6426 | Buclizine dihydrochloride | Longifene,Buclina,Buclizine HCl,UCB-4445 | 5-HT Receptor , AChR , Histamine Receptor |
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ... | |||
T68068 | Ezlopitant | CJ 11974,CJ-11974,CJ11974 | Neurokinin receptor |
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain. | |||
T68068L | (R)-CJ 11974 | Neurokinin receptor | |
(R)-CJ 11974 is a novel non-peptide neurokinin NK1 substance P receptor antagonist with potential analgesic activity that can be used to study chemotherapy-induced vomiting. | |||
T1156 | Palonosetron hydrochloride | RS 25259 197,Palonosetron HCl,RS 25259 | 5-HT Receptor |
Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting. | |||
T6616 | Ondansetron hydrochloride | SN 307,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran | 5-HT Receptor |
Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation therapy. | |||
T4568 | Dolasetron | MDL-73147 | 5-HT Receptor |
Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy. | |||
T5009 | Trimethobenzamide hydrochloride | Ro 2-9578,Tribenzagan Hydrochloride | Dopamine Receptor , Influenza Virus |
Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. |