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Clebopride malate

Catalog No. T7569 CAS 57645-91-7

Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.

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Clebopride malate, CAS 57645-91-7

Pack Size	Availability	Price/USD
5 mg	In stock	$ 47.00
10 mg	In stock	$ 67.00
25 mg	In stock	$ 106.00
50 mg	In stock	$ 147.00
100 mg	In stock	$ 247.00
200 mg	In stock	$ 368.00
1 mL * 10 mM (in DMSO)	In stock	$ 53.00

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Purity: 99.97%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.
In vivo	Clebopride, a new benzamide derivative, has, in common with the other members of this group,and with antiemetic drug, antidopaminergic activity.?In animals, its therapeutic ratio is superior to that of metoclopramide at doses free of side effects associated with hyperprolactinemia and extrapyramidal symptoms[1].

Molecular Weight	507.96
Formula	C24H30ClN3O7
CAS No.	57645-91-7

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 34 mg/mL (66.93 mM)

References and Literature

1. Bleiberg H , Piccart M , Lips S , et al. A phase I trial of a new antiemetic drug--clebopride malate--in cisplatin-treated patients[J]. Annals of Oncology Official Journal of the European Society for Medical Oncology, 1992, 3(2):141. 2. Kawasaki H , Yamamoto M , Okayasu H , et al. [A case of respiratory dyskinesia due to clebopride malate][J]. Rinsho shinkeigaku = Clinical neurology, 1991, 31(8):878-881.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Anti-Cancer Drug Library Drug Repurposing Compound Library Anti-Neurodegenerative Disease Compound Library GPCR Compound Library Anti-Cancer Approved Drug Library Anti-Parkinson's Disease Compound Library Bioactive Compounds Library Max Neurotransmitter Receptor Compound Library FDA-Approved & Pharmacopeia Drug Library

Related Products

Related compounds with same targets

Acetophenazine dimaleate Nomifensine GBR 12935 dihydrochloride Molindone NEO 376 Tetrabenazine PG 01037 dihydrochloride Tolnapersine TFA

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Keywords

Clebopride malate 57645-91-7 GPCR/G Protein Neuroscience Dopamine Receptor Clebopride Inhibitor inhibit Clebopride Malate inhibitor

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