11
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T20720 | Norethisterone enanthate | NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564 | Estrogen/progestogen Receptor |
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects. | |||
T1490 | Gestodene | SHB 331,WL 70 | Estrogen/progestogen Receptor , Progesterone Receptor |
Gestodene (WL 70) is a progestogen hormonal contraceptive. | |||
T0870 | Altrenogest | R2267,RU2267,Allyltrenbolone,A35957 | Estrogen/progestogen Receptor , Progesterone Receptor |
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone. | |||
T3036 | Dydrogesterone | Progesterone Receptor | |
Dydrogesterone is a potent progestogen which can be used in progesterone deficiency studies. | |||
T0301 | Ethisterone | 17α-Ethynyltestosterone,Pregneninolone | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone. | |||
T2577 | Dienogest | STS 557 | Apoptosis , Estrogen/progestogen Receptor , Progesterone Receptor , Autophagy |
Dienogest (STS 557) is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic activities that is used in hormone therap... | |||
T1284 | Megestrol acetate | SC10363,BDH1298 | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , HIV Protease , Autophagy |
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. It is given by mouth in the palliative treatment ... | |||
T0272 | Nilutamide | RU23908 | Androgen Receptor |
Nilutamide (RU23908), an antineoplastic hormonal agent, is mainly used in the treatment of prostate Y. Nilutamide is a pure, nonsteroidal anti-androgen with affinity for androgen receptors, but not for estrogen, progesto... | |||
T25429 | Flumedroxone acetate | WG 537,NSC 52412,NSC-52412,NSC52412,Leomigran | |
Flumedroxone acetate is a progestogen medication which is or has been used as an antimigraine. | |||
T20755 | Trimegestone | RU27987,RU-27987,RU 27987 | |
Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation. | |||
T25304 | Demegestone | R-2453,Lutionex,R 2453,RU 2453,R2453 | |
Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat lutea... |