antimuscarinic — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T9353	OXOMEMAZINE		AChR , Histamine Receptor
	Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...		AChR , Histamine Receptor
T8383	Cyclopentolate Hydrochloride		AChR
	Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.		AChR
T5023	Propiverine hydrochloride		Others , Calcium Channel , AChR
	Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).		Others , Calcium Channel , AChR
T9419	Fesoterodine	(R) Fesoterodine	AChR
	Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB).		AChR
T0786	Clidinium bromide	Ro 2-3773	AChR
	Clidinium bromide (Ro 2-3773) , a synthetic anticholinergic agent, has been shown in experimental and clinical researchers to have a pronounced antisecretory and antispasmodic effect on the gastrointestinal tract. It can...		AChR
T1475	Fesoterodine fumarate	Toviaz,SPM 907	AChR
	Fesoterodine fumarate (Toviaz) is the fumarate salt form of fesoterodine, a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. Fesoterodine is rapidly hydrolyzed in vivo...		AChR
T0862	Diphenidol hydrochloride	Diphenidol HCl,Difenidol hydrochloride	Sodium Channel , AChR
	Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.		Sodium Channel , AChR
T2138	Oxyphencyclimine Hydrochloride	Spazamin,Daricon,Ulcociclinina	AChR
	Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.		AChR
T1474	Otilonium bromide	Octylonium bromide,SP63	Calcium Channel , AChR
	Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.		Calcium Channel , AChR
T7002	Trihexyphenidyl hydrochloride	Triesifenidile,Benzhexol hydrochloride,Tremin,Artane hydrochloride	AChR
	Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.		AChR
T7555	Piperidolate hydrochloride		AChR
	Piperidolate hydrochloride is an antimuscarinic, could restrain the abnormal activity caused by acetylcholine. inhibits intestinal cramp induced by acetylcholine (rats and dogs).		AChR
T0427	Homatropine Methylbromide	Homatropine methobromide	AChR
	Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.		AChR
T2222	Carbinoxamine Maleate Salt	Lergefin,CarbinoxaMine Maleate	Histamine Receptor
	Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.		Histamine Receptor
T9420	Prifinium bromide		Others
	Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.		Others
T9877	Tiquizium		AChR
	Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.		AChR
T1197	Trimebutine maleate	Debridat,Polibutin	Calcium Channel , Opioid Receptor
	Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate receptors served as a spasmolytic drug for therapy of both c...		Calcium Channel , Opioid Receptor
T0918	Trimebutine	Mebutin	Opioid Receptor
	Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid agonist effects. It is marketed for the treatment of irritabl...		Opioid Receptor
T67956L	Litoxetine HCl	litoxetine HCL(86811-09-8 Free base)	5-HT Receptor
	Litoxetine HCl is a selective 5-hydroxytryptamine (5-HT) reuptake inhibitor (SSRI) and mixed 5-hydroxytryptamine antagonist used in the treatment of urinary incontinence. Litoxetine HCl in the absence of antimuscarinic c...		5-HT Receptor
T28523	Revatropate	UK-112 166,UK 112166,UK-112,166
	Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.
T11275	Fesoterodine L-mandelate		Others
	Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).		Others