trap-1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T7625	TRAP-6	PAR-1 agonist peptide,Thrombin Receptor Activator Peptide 6,TRAP-6(2TFA)	Protease-activated Receptor
	TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).		Protease-activated Receptor
TP1015	NFAT Inhibitor	VIVIT peptide	Others
	NFAT Inhibitor (VIVIT peptide) is a cell-permeable compound that selectively inhibits calcineurin-mediated dephosphorylation of NFAT.		Others
T8958	PU-H54		GPR
	PU-H54 is a purine-based inhibitor of Grp94. It is a Grp94-selective resorcinol-based inhibitor isolated through probing of the exclusive binding region of S2 subpocket in Grp94.		GPR
T60557	TRAP-6-IN-1
	TRAP-6-IN-1 (Compound 8) is a dual inhibitor of collagen and TRAP-6 with IC 50 values of 17.12 μM and 11.88 μM, respectively. TRAP-6-IN-1 non-competitively inhibits agonist-induced platelet aggregation[1].
T38852L	TRAP-6 amide acetate		Protease-activated Receptor
	TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].		Protease-activated Receptor
T2114	VER-82576	NVP-BEP800	HSP
	VER-82576 (NVP-BEP800), a synthetic HSP90β inhibitor (IC50: 58 nM), exhibits >70-fold selectivity against Hsp90 family members Trap-1 and Grp94.		HSP
T38961L	DP-1 hydrochloride	DP-1 hydrochloride(1472616-61-7 Free base)	Drug Metabolite
	DP-1 hydrochloride is a degradation product of SDC-TRAP-0063, a fragment of Ganetespib, a heat shock protein 90 (HSP90) inhibitor with antitumor activity.		Drug Metabolite
T22739	DMPO	5,5-Dimethyl-1-pyrroline N-oxide	Others
	DMPO (5,5-Dimethyl-1-pyrroline N-oxide) is a kind of water-soluble nitric oxide spin trap, which allows the measurement of oxygen-centered free radicals in biological systems at room temperature using electron spin reson...		Others
T3098	Vorapaxar sulfate	SCH 530348 sulfate,Zontivity,vorapaxar monosulfate	Protease-activated Receptor
	Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.		Protease-activated Receptor
T7013	Vorapaxar	SCH 530348,MK-5348	Protease-activated Receptor
	Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).		Protease-activated Receptor
T38887	TRAP-6 amide TFA
	TRAP-6 amide TFA is a PAR-1 thrombin receptor agonist peptide.
T80111	TRAP-5 amide
	TRAP-5 amide is a peptide agonist for protease-activated receptor 1 (PAR 1) [1].
T38852	TRAP-6 amide
	TRAP-6 amide is a PAR-1 thrombin receptor agonist peptide.
T80108	Hepcidin-1 (mouse)
	Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion. This compound also reduces FPN1 protein levels and boosts intra...
T78099	Iso-TRAP-6	iso-SFLLRN
	Iso-TRAP-6 (iso-SFLLRN) is an analog of TRAP-6 and a PAR-1 agonist, utilizing isoserine in place of serine as the first amino acid, and is capable of activating platelets [1].
T78037	Hepcidin-1 (mouse) TFA
	Hepcidin-1 (mouse) TFA, an endogenous peptide hormone, regulates iron homeostasis by upregulating mRNA levels of TRAP, cathepsin K, and MMP-9, enhancing TRAP-5b protein secretion, and downregulating FPN1 protein levels, ...
T7496	Thrombin Receptor Activator for Peptide 5 (TRAP-5)	Thrombin Receptor Activator for Peptide	Protease-activated Receptor
	Thrombin Receptor Activator for Peptide 5 (TRAP-5), also known as Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), is employed in coronary heart disease (CHD) research.		Protease-activated Receptor
T38961	DP-1
	DP-1, a Ganetespib degradation product, represents a fragment derived from SDC-TRAP-0063. Ganetespib itself functions as an inhibitor of heat shock protein 90 (HSP90), exhibiting notable anti-tumor properties.
T36777	Thrombin Receptor Agonist Peptide (trifluoroacetate salt)
	Thrombin receptor agonist peptide (TRAP-14) is a 14-amino acid peptide agonist of the α-thrombin receptor. It induces aggregation of washed platelets as well as platelets in citrated and hirudin plasma. TRAP-14 (100 μM) ...
T35867	TRAP-6 Peptide (trifluoroacetate salt)
	TRAP-6 peptide is a hexapeptide corresponding to residues 42-47 of protease-activated receptor 1 (PAR1). It acts as an agonist of PAR1, inducing platelet aggregation in human platelet-rich plasma ex vivo (EC50 = 0.8 μM)....