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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T84293 | SSR 180 | ||
T28855 | SSR126768A | SSR-126768A,SSR 126768A | Oxytocin Receptor |
SSR126768A is a novel and selective, orally active and potent oxytocin (OT) receptor antagonist with inhibitory effects on uterine contractions for the prevention of preterm labor. | |||
T6082 | SSR128129E | SSR | FGFR |
SSR128129E (SSR) is an allosteric and orally-active FGFR1 inhibitor (IC50: 1.9 μM), but not affecting other related RTKs. | |||
T31095 | Crinecerfont | SSR125543,SSR 125543,SSR-125543,SSR125543A,SSR 125543A,SSR-125543A | CRFR |
Crinecerfont (SSR-125543) is a selective antagonist of corticotropin-releasing factor 1 receptor (CRF1) and can be used in studies about Classic congenital adrenal hyperplasia. | |||
T69140 | Burapitant | SSR 240600 | Neurokinin receptor |
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity. | |||
T28857 | SSR-182289A (Free) | SSR182289,SSR-182289A,SSR-182289,SSR 182289A,SSR182289A,SSR 182289 | |
SSR-182289A (Free) is a thrombin inhibitor. | |||
T28856 | SSR180711 hydrochloride | SSR-180711A HCl,SSR-180711C HCl,SR-180711 HCl | AChR |
SSR180711 hydrochloride (SSR-180711A HCl) is a selective Alpha7 nicotinic acetylcholine partial agonist for the study of neurodegenerative and cognitive disorders. | |||
T21989 | SSR 69071 | ||
SSR69071 is a potent, orally active, and selective inhibitor of neutrophil elastase. SSR69071 displays a higher affinity for human elastase (Ki =0.0168 nM) than for rat (Ki =3 nM), mouse (Ki =1.8 nM), and rabbit (Ki = 58... | |||
T13002 | SSR-241586 | Others | |
SSR-241586 is a neurokinin receptors antagonist,and is shown to be active in the treatment of depression, schizophrenia, urinary trouble, emesis, and irritable bowel syndrome (IBS). | |||
T23395 | SSR 146977 hydrochloride | Others | |
NK3 receptor antagonist | |||
T5048 | SSR240612 | Bradykinin Receptor | |
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively). | |||
T28858 | SSR504734 | SSR-504734,SSR 504734 | |
SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor. | |||
T40398 | Crinecerfont hydrochloride | SSR-125543A,SSR-125543 hydrochloride | |
Crinecerfont hydrochloride (SSR-125543) is a highly potent, orally active, non-peptide antagonist of the CRF1 receptor. It has demonstrated efficacy in the context of Classic congenital adrenal hyperplasia (CAH) research... | |||
T13003 | SSR128129E free acid | SSR free acid | FGFR |
SSR128129E free acid is an orally available and allosteric inhibitor of FGFR(IC50 of 1.9 μM for FGFR1). | |||
T15276 | Ferroquine | SSR97193,Ferrochloroquine | Others |
Ferroquine (Ferrochloroquine) is a ferrocenyl analogue of Chloroquine with antimalarial activity. Ferroquine induces oxidative stress and the subsequent destruction of the membrane, resulting in parasiticidal effect on P... | |||
T28153 | Nelivaptan | SSR149415,SR 149415,SR-149415 | Vasopressin Receptor |
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist. | |||
T40775 | SSR411298 | SSR411298 | |
SSR411298 is a reversible, orally active compound that selectively inhibits fatty acid amide hydrolase (FAAH). Its potential lies in the field of post-traumatic stress disorder (PTSD) research. | |||
T11006 | Desmethyl ferroquine | SSR97213 | Others |
Desmethyl ferroquine is the active and major metabolite of Ferroquine.Desmethyl ferroquine shows significant activity against Chloroquine-susceptible and resistant P. falciparum strains. Ferroquine is an antimalarial. | |||
T90597 | SSR504734 HCl | ||
SSR504734 is an orally active, selective and reversible inhibitor of human, rat, and mouse GlyT1 ( IC 50 =18, 15, and 38 nM, respectively). SSR504734 exhibits activity in schizophrenia, anxiety and depression models [1]. | |||
T60126 | 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine | Others , CRFR | |
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine is an enantiomeric counterpart of SSR-125543. SSR-125543 is a potent CRF-R1 antagoni... |