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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0468 | Lidocaine | Lignocaine,Alphacaine,Xylocaine | Apoptosis , ERK , NF-κB , MEK , Sodium Channel , Histamine Receptor |
Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation of intracellular adhesion molecule-1 (ICAM-1), pro-inflammat... | |||
T1144 | Lidocaine hydrochloride | Lidocaine HCL,Lignocaine hydrochloride,Xyloneural,Lidothesin | Apoptosis , ERK , NF-κB , MEK , Sodium Channel |
Lidocaine hydrochloride (Lignocaine hydrochloride) is a local anesthetic and cardiac depressant used as an antiarrhythmic agent. Its actions are more intense and its effects more prolonged than those of PROCAINE but its ... | |||
T1144L | Lidocaine Hydrochloride hydrate | EGFR , Sodium Channel | |
Lidocaine Hydrochloride hydrate is an amide local anesthetic, has anti-inflammatory property. | |||
T25720 | Lidocaine methiodide | Methyllidocaine iodide,N-Methyllidocaine | |
Lidocaine methiodide is an antiarrythmic. It is also exhibiting arrythmogenic effects in subjects. | |||
T23213 | QX-222 chloride | QX 222,Lidocaine N-Methyl Hydrochloride | Sodium Channel |
QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker. | |||
T8341 | QX 314 | QX-314 | Others |
QX 314 (Lidocaine N-ethyl bromide) is a blocker of non-membrane-permeable,and Inhibits Acid-Induced Activation of Esophageal Nociceptive C Fiber Neurons. | |||
T13177L | Tocainide | Sodium Channel | |
Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus. | |||
T10679 | Carcainium chloride | QX 572,Carcainium (chloride),Carcainiumchloride,RSD 931 | Others |
Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect. | |||
T26287 | Transcainide | R54718,R 54718,R-54718 | Sodium Channel |
Transcainide(R 54718), a new lidocaine analog, is an orally active antiarrhythmic agent.Transcainide blocks the open state of BTX-activated sodium channels in bovine heart and rat skeletal muscle. | |||
T9530 | W 36017 | Others | |
W36017 is an impurity of lidocaine with a PKA of 7.4 for blocking neurologic activity. | |||
T13177 | Taquidil | ||
Tocainide hydrochloride is a sodium channel blocker, it blocks the sodium channels in the pain-producing foci in the nerve membranes. Tocainide hydrochloride is an orally effective antiarrhythmic agent, structurally and ... | |||
T1098 | Denatonium benzoate | THS-839 | Others |
Denatonium benzoate (THS-839) , a quaternary ammonium cation, is a compound of a salt with an inert anion like saccharide or benzoate. Its structure is involved in the local anesthetic lidocaine which difference only is ... | |||
T34253 | Rad 242 | Rad242,Rad-242 | |
Rad 242 is a hydrophobic lidocaine derivative. | |||
T30861 | CH 200 | CH-200,CH200,06-14C | |
CH 200 is a novel antiarrhythmic drug that inhibits arrhythmias in beagles more effectively than procainamide and lidocaine. | |||
T20732 | Lignocaine N-oxide | ||
Lignocaine N-oxide is a metabolite of Lidocaine, which is an antiarrhythmic and anesthetic agent. | |||
T80638 | Glycinexylidide | GX | MEK |
Glycinexylidide (GX), the active metabolite of the local anesthetic Lidocaine, exhibits properties significant in inhibiting sodium channels with complex voltage dependence and mitigates the proliferation and spread of g... | |||
T37670 | CAY10568 | ||
Most local anesthetics act by abolishing voltage gated sodium channel currents indiscriminately in all populations of neurons. Selective analgesia through TRPV1-mediated entry of a cationic lidocaine derivative, QX314, w... |