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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T17103 | TM-N1324 | Others , GHSR | |
TM-N1324 is a GPR39 agonist. TM-N1324 activates human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively. TM-N1324 has similar potencies to murine GPR39 with EC50s... | |||
T4648 | TC-G-1008 | GPR39-C3 | GHSR |
TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively). | |||
TQ0022 | Capromorelin Tartrate | CP 424391-18 | GHSR |
Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a). | |||
T16508 | PF-5190457 | PF-05190457 | GHSR |
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36). | |||
T10319 | Anamorelin | RC-1291,ONO-7643 | GHSR |
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). | |||
T7112 | Ibutamoren Mesylate | MK-0677,MK-677 | GHSR |
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist. | |||
T7225 | AnaMorelin hydrochloride | RC-1291 hydrochloride,ONO-7643 hydrochloride | GHSR |
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay). | |||
T34281 | Relamorelin | BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131 | GHSR |
Relamorelin (RM-131), a selective and potent growth hormone-releasing peptide/growth hormone secretagogue receptor (GHSR) agonist, is a potent growth hormone-releasing peptide mimetic with a high affinity for the GHS-1a ... | |||
T31734 | BMS-604992 | EX1314,EX-1314 HCl,EX-1314,BMS604992,EX-1314 hydrochloride, BMS-604992,EX 1314 | |
EX-1314 (BMS-604992) is a growth hormone secretagogue receptor (GHSR) agonist. | |||
T38959 | BMS-604992 dihydrochloride | EX-1314 dihydrochloride,BMS-604992 dihydrochloride | |
BMS-604992 (EX-1314) dihydrochloride is a selective and orally active small-molecule agonist of the growth hormone secretagogue receptor (GHSR). It exhibits high-affinity binding (k i = 2.3 nM) and potent functional acti... | |||
T40876 | BMS-604992 free base | BMS-604992 free base,EX-1314 free base | |
BMS-604992 (EX-1314) free base is a selective, orally active small-molecule growth hormone secretagogue receptor (GHSR) agonist. It exhibits high-affinity binding (k i = 2.3 nM) and potent functional activity (EC 50 = 0.... | |||
T28812 | SM-130686 | SM 130686,SM130,686,SM 130,686 | |
SM-130,686 is a potent, orally-active agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and growth hormone secretagogue. It has around half the potency of the endogenous agonist ghrelin as a stimulator o... | |||
T68276 | Macimorelin acetate | EP-1572 acetate ; AEZS-130 acetate,AEZS-130 acetate,EP-1572 acetate | |
Macimorelin Acetate (EP-1572), an orally active growth hormone (GH) secretagogue and a ghrelin receptor (GHSR) agonist, stimulates GH release. It is utilized in research focusing on adult growth hormone deficiency (AGHD)... | |||
T76318 | GHRF, porcine | ||
GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing the release of growth hormone [1] [2]. | |||
T75262 | Relamorelin TFA | ||
Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, acts as a potent and selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR), with a K_i of 0.42 nM for the GHS-1a receptor. This compound is... | |||
T39236 | Relamorelin acetate | Relamorelin acetate,RM-131 acetate,BIM-28131acetate | |
Relamorelin (RM-131) acetate is a pentapeptide ghrelin analog that acts as a selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR). It exhibits a high affinity for the GHS-1a receptor, with a Ki v... |