dp1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T38961	DP-1
	DP-1, a Ganetespib degradation product, represents a fragment derived from SDC-TRAP-0063. Ganetespib itself functions as an inhibitor of heat shock protein 90 (HSP90), exhibiting notable anti-tumor properties.
T38961L	DP-1 hydrochloride	DP-1 hydrochloride(1472616-61-7 Free base)	Drug Metabolite
	DP-1 hydrochloride is a degradation product of SDC-TRAP-0063, a fragment of Ganetespib, a heat shock protein 90 (HSP90) inhibitor with antitumor activity.		Drug Metabolite
T4297	Flibanserin	BIMT-17BS,Girosa,BIMT-17	Dopamine Receptor , 5-HT Receptor
	Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. Flibanserin has been associated with a low rate of minor serum aminotransferase elevations during treatment but has n...		Dopamine Receptor , 5-HT Receptor
T78033	SDP116
	SDP116, a synthetic peptide derivative of the GPR116 Stachel sequence, exhibits ADGRF5 agonistic activity [1].
TN2358	Fructo-oligosaccharide DP10/GF9	Fructo-oligosaccharide DP10/GF9	Others
	Fructo-oligosaccharide DP10/GF9 is a compound classified as a fructooligosaccharide (FOS) with a degree of polymerization (DP) of 10. FOS consists of a chain of 9 fructose units connected by (2→1)-β-glycosidic bonds, wit...		Others
T76219	MDP1
	MDP1, derived from Melittin, disrupts the membrane integrity of both Gram-positive and Gram-negative bacteria, leading to bacterial death through membrane damage. This compound exhibits potent antibacterial activity agai...
T19328	Fructo-oligosaccharide DP11/GF10		Others
	Fructo-oligosaccharide DP11/GF10 is a fructooligosaccharide (FOS) compound with a degree of polymerization (DP) equal to 11. FOS consists of 10 fructose units connected by (2→1)-β-glycosidic bonds, with a single D-glucos...		Others
T76219L	MDP1 acetate
	MDP1 acetate, a derivative of Melittin, compromises the membrane integrity of both Gram-positive and Gram-negative bacteria leading to bacterial death through membrane damage. It exhibits potent antibacterial activity ag...
T82369	Fructo-oligosaccharide DP14
	Fructo-oligosaccharide DP14, an oligosaccharide derived from Atractylodes lancea [1], represents a specific polysaccharide subclass with a degree of polymerization of 14.
T82370	Fructo-oligosaccharide DP13
	Fructo-oligosaccharide DP13 is an inulin-type fructan that can be isolated from Morinda officinalis [1].
T19329	Fructo-oligosaccharide DP12/GF11		Others
	Fructo-oligosaccharide DP12/GF11 is a member of fructooligosaccharides (FOS) characterized by a degree of polymerization (DP) of 12. FOS compounds consist of 11 fructose units connected by (2→1)-β-glycosidic bonds, with ...		Others
T13109	TDP1 Inhibitor-1		Others
	TDP1 Inhibitor-1 is a potent inhibitor of Tyrosyl-DNA Phosphodiesterase 1 (TDP1) (IC50 of 7 μM).		Others
T62965	TDP1 Inhibitor-2
	TDP1 Inhibitor-2 is a potent inhibitor of TDP1 (tyrosyl-DNA phosphodiesterase 1) (IC50: 99 nM) and inhibits SCAN1 (spinal cerebellar ataxia syndrome with axonal neuropathy) (IC50: 3.5 μM).
T5386	Asapiprant		Prostaglandin Receptor
	Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.		Prostaglandin Receptor
T5150	Treprostinil	LRX-15,Orenitram,Remodulin	Prostaglandin Receptor
	Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).		Prostaglandin Receptor
T14842	BW 245C	BW245C	Prostaglandin Receptor
	BW 245C is a selective prostaglandin-like DP receptor (DP1) agonist, a prostaglandin analogue with inhibitory effects on the aggregation response of collagen, which can be used to study diseases such as stroke.		Prostaglandin Receptor
T15712	Laropiprant	MK-0524	Prostaglandin Receptor
	Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki = 2.95 nM).		Prostaglandin Receptor
T4635	Ralinepag	APD811	Others , Prostaglandin Receptor
	Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.		Others , Prostaglandin Receptor
T5171	Treprostinil Sodium	UT-15	VEGFR , c-RET , Prostaglandin Receptor
	Treprostinil Sodium (UT-15) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).		VEGFR , c-RET , Prostaglandin Receptor
T63349	Treprostinil diethanolamine	UT-15C	Prostaglandin Receptor
	Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1, EP4, EP3 and FPKi, respectively. Treprostinil diethanolamine i...		Prostaglandin Receptor