Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against δPI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, β, and γ).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 233.00 | |
2 mg | In stock | $ 346.00 | |
5 mg | In stock | $ 583.00 | |
10 mg | In stock | $ 835.00 | |
25 mg | In stock | $ 1,270.00 | |
50 mg | In stock | $ 1,690.00 | |
100 mg | In stock | $ 2,290.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 826.00 |
Description | Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against δPI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, β, and γ). |
Synonyms | TGR-1202 R-enantiomer, RP5264 R-enantiomer |
Molecular Weight | 571.55 |
Formula | C31H24F3N5O3 |
CAS No. | 1532533-69-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 9 mg/mL (15.75 mM)
You can also refer to dose conversion for different animals. More
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Umbralisib R-enantiomer 1532533-69-9 PI3K/Akt/mTOR signaling PI3K TGR-1202 R-enantiomer RP5264 R-enantiomer inhibitor inhibit