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Tamsulosin

Catalog No. T0210L CAS 106133-20-4

Synonyms: LY253351 free base, HSDB7744, (R)-(-)-YM12617 free base, Harnal-D, Flowmax, HSDB 7744, HSDB-7744

Tamsulosin ((R)-(-)-YM12617 free base) is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulosin is used to treat difficulty urinating, a common symptom of an enlarged prostate. Tansulosin and other drugs called alpha blockers work by relaxing the neck muscles of the bladder and muscle fibers in the prostate itself, making it easier to urinate.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Tamsulosin, CAS 106133-20-4

Pack Size	Availability	Price/USD
5 mg	In stock	$ 30.00
10 mg	In stock	$ 47.00
25 mg	In stock	$ 73.00
50 mg	In stock	$ 97.00
100 mg	In stock	$ 147.00
1 mL * 10 mM (in DMSO)	In stock	$ 52.00

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Purity: 99.94%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	LY253351 free base, HSDB7744, (R)-(-)-YM12617 free base, Harnal-D, Flowmax, HSDB 7744, HSDB-7744
Molecular Weight	408.51
Formula	C20H28N2O5S
CAS No.	106133-20-4

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 90.0 mg/mL (220.3 mM), Sonication is recommended.

References and Literature

1. Özsoy M, Liatsikos E, Scheffbuch N, Kallidonis P. Comparison of silodosin to tamsulosin for medical expulsive treatment of ureteral stones: a systematic review and meta-analysis. Urolithiasis. 2016 Mar 28. 2. Dimitropoulos K, Gravas S. Fixed-dose combination therapy with dutasteride and tamsulosin in the management of benign prostatic hyperplasia. Ther Adv Urol. 2016 Feb;8(1):19-28. 3. Dimitropoulos K, Gravas S. Solifenacin/tamsulosin fixed-dose combination therapy to treat lower urinary tract symptoms in patients with benign prostatic hyperplasia. Drug Des Devel Ther. 2015 Mar 19;9:1707-16. 4. Shim SR, et al. General effect of low-dose tamsulosin (0.2 mg) as a first-line treatment for lower urinary tract symptoms associated with benign prostatic hyperplasia: a systematic review and meta-analysis. Curr Med Res Opin. 2015 Feb;31(2):353-65.

Related compound libraries

This product is contained In the following compound libraries：

Anti-Cancer Drug Library Anti-Cancer Approved Drug Library GPCR Compound Library Membrane Protein-targeted Compound Library Drug Repurposing Compound Library Anti-Cancer Clinical Compound Library Approved Drug Library Bioactive Compound Library Neuronal Signaling Compound Library Anti-Cancer Compound Library

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Related compounds with same targets

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Tamsulosin 106133-20-4 GPCR/G Protein Neuroscience Adrenergic Receptor LY253351 free base LY253351 HSDB7744 YM-12617 (R)-(-)-YM12617 free base YM12617 YM 12617 Harnal-D Flowmax YM12617 free base LY-253351 HSDB 7744 LY 253351 HSDB-7744 inhibitor inhibit

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