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TRPM8 antagonist WS-3

Catalog No. T5962 CAS 39711-79-0

Synonyms: Cyclohexanecarboxamide, N-Ethyl-p-menthane-3-carboxamide, N-Ethyl-2-isopropyl-5-methylcyclohexanecarboxamide

TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).

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TRPM8 antagonist WS-3 Chemical Structure

TRPM8 antagonist WS-3, CAS 39711-79-0

Pack Size	Availability	Price/USD	Quantity
1 g	In stock	$ 30.00
1 mL * 10 mM (in DMSO)	In stock	$ 29.00

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM).
Targets&IC50	TRPM8:3.7 μM (EC50)

Synonyms	Cyclohexanecarboxamide, N-Ethyl-p-menthane-3-carboxamide, N-Ethyl-2-isopropyl-5-methylcyclohexanecarboxamide
Molecular Weight	211.34
Formula	C13H25NO
CAS No.	39711-79-0

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 100 mg/mL (473.17 mM)

References and Literature

1. H‐J Behrendt, Germann T , Gillen C , et al. Characterization of the mouse cold‐menthol receptor TRPM8 and vanilloid receptor type‐1 VR1 using a fluorometric imaging plate reader (FLIPR) assay[J]. British Journal of Pharmacology, 2004, 141(4).

Related compound libraries

This product is contained In the following compound libraries：

Membrane Protein-targeted Compound Library NO PAINS Compound Library Bioactive Compound Library Food Additive Library Human Endogenous Metabolite Compound Library Plus Ion Channel Inhibitor Library Anti-Cancer Compound Library Bioactive Compounds Library Max Human Metabolite Library Neuronal Signaling Compound Library

Related Products

Related compounds with same targets

AP 18 Linoleoyl Ethanolamide OMDM-5 ICILIN SET 2 M8-B Hydrochloride JT010 RQ-00203078

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Keywords

TRPM8 antagonist WS-3 39711-79-0 Membrane transporter/Ion channel TRP/TRPV Channel TRP Channel inhibit TRPM8 antagonist WS3 Cyclohexanecarboxamide TRPM8 agonist WS-3 N-Ethyl-p-menthane-3-carboxamide N-Ethyl-2-isopropyl-5-methylcyclohexanecarboxamide Transient receptor potential channels TRPM-8 antagonist WS-3 TRPM8 antagonist WS 3 Inhibitor inhibitor

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