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Prilocaine

Catalog No. T6953 CAS 721-50-6

Synonyms: NSC 40027, Propitocaine, Citanest, Propitocaine, Citanest NSC 40027

Purity 99.67% Datasheet

Prilocaine is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of seizures.

Prilocaine, CAS 721-50-6

Pack Size	Availability	Price/USD
25 mg	In stock	50.00
50 mg	In stock	81.00
100 mg	In stock	120.00
200 mg	In stock	217.00
1 mL * 10 mM (in DMSO)	In stock	69.00

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Purity 99.67%

HNMR HPLC COA Datasheet MSDS

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Prilocaine is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of seizures.
Targets&IC50	Sodium Channel,

Synonyms	NSC 40027 , Propitocaine , Citanest , Propitocaine , Citanest NSC 40027
Purity	99.67%
Molecular Weight	220.31
Formula	C13H20N2O
CAS No.	721-50-6

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

DMSO: 41 mg/mL (186.1 mM)

Ethanol: 41 mg/mL (186.1 mM)

Water: <1 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Eriksson E. Prilocaine. Acta Chir Scand Suppl. 1966;358:1-82. 2. Juhlin L, et al. EMLA: a new topical anesthetic. Adv Dermatol. 1990;5:75-91; discussion 92.

Related compound libraries

This product is contained In the following compound libraries：

Approved Drug Library Bioactive Compound Library Ion Channel Inhibitor Library FDA-approved Drug Library

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Related compounds with same targets

Karanjin Hexamethylene amiloride EIPA Pilsicainide HCl Fosphenytoin sodium Ibutilide Fumarate Actein Ralfinamide mesylate

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
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Tech Support

Answers to questions you may have can be found in the Inhibitor Handling Instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.