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Mirogabalin

Name: Mirogabalin
Brand: TargetMol
SKU: T7216
Price: 35 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T7216Cas No. 1138245-13-2

Alias DS5565

Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.

Mirogabalin

🥰Excellent

Purity: 98.57%

Catalog No. T7216Alias DS5565Cas No. 1138245-13-2

Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.

Pack Size	Price	Availability
1 mg	$35	In Stock
5 mg	$81	In Stock
10 mg	$127	In Stock
25 mg	$222	In Stock
50 mg	$338	In Stock
100 mg	$513	In Stock
500 mg	$1,080	In Stock

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Purity:98.57%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.
In vivo	Mirogabalin has potent and sustained analgesic effects (ED50 = 2.5 mg/kg) in rats with diabetes induced by streptozotocin .?Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50 = 9.4 mg/kg) or locomotor activity (ID50 = 43.9 mg/kg), at its effective dose.
Synonyms	DS5565

Chemical Properties

Molecular Weight	209.28
Formula	C₁₂H₁₉NO₂
Cas No.	1138245-13-2
Smiles	CCC1=C[C@@H]2[C@@H](C[C@]2(CN)CC(O)=O)C1
Relative Density.	1.104 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 1.83 mg/mL (8.76 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	4.7783 mL	23.8914 mL	47.7829 mL	238.9144 mL
5 mM	0.9557 mL	4.7783 mL	9.5566 mL	47.7829 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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