Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 38.00 | |
5 mg | In stock | $ 61.00 | |
10 mg | In stock | $ 101.00 | |
25 mg | In stock | $ 207.00 | |
50 mg | In stock | $ 328.00 | |
100 mg | In stock | $ 531.00 | |
500 mg | In stock | $ 1,180.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 68.00 |
Description | GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites. |
Targets&IC50 | D3:ki:0.4 nM |
In vitro | GR 103691 shows a marked affinity for α-1 adrenoceptors (Ki: 12.6 nM) and serotonin1A (5-HT1A) receptors (Ki: 5.8 nM). |
Molecular Weight | 485.62 |
Formula | C30H35N3O3 |
CAS No. | 162408-66-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.86 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
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GR 103691 162408-66-4 GPCR/G Protein Neuroscience Dopamine Receptor Inhibitor GR-103691 GR103691 inhibit inhibitor