Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 166.00 | |
5 mg | In stock | $ 331.00 | |
10 mg | In stock | $ 563.00 | |
25 mg | In stock | $ 887.00 | |
50 mg | In stock | $ 1,230.00 | |
100 mg | In stock | $ 1,670.00 | |
500 mg | In stock | $ 3,330.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 535.00 |
Description | Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction. |
Targets&IC50 | Aortic contraction:0.8 μM , Aortic contraction:0.8 μM |
In vivo | Calcium channel-modulator-1 (20 mg/kg ; p.o.) causes a 35-37% decrease in systolic blood pressure in spontaneously hypertensive rats. However, iv administration of Calcium channel-modulator-1 to anesthetized spontaneously hypertensive rats causes a decrease in blood pressure.[1] |
Molecular Weight | 579.45 |
Formula | C26H24Cl2N2O7S |
CAS No. | 136941-70-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.79 mg/mL (10 mM), Sonification is recommended
You can also refer to dose conversion for different animals. More
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Calcium channel-modulator-1 136941-70-3 Membrane transporter/Ion channel Metabolism Others Calcium Channel Calcium channelmodulator1 Calcium channel modulator 1 inhibitor inhibit