Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 95.00 | |
2 mg | In stock | $ 143.00 | |
5 mg | In stock | $ 219.00 | |
10 mg | In stock | $ 329.00 | |
25 mg | In stock | $ 562.00 | |
50 mg | In stock | $ 790.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 222.00 |
Description | Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase. |
Targets&IC50 | DPPH:54.53 ug/mL, Anti-plasmodial:5.80 μM |
In vitro | Atherosperminine shows strong anti-plasmodial activity against Plasmodium falciparum, with the IC50 value of 5.80 μM. Atherosperminine also shows antioxidant activity in a DPPH assay with the IC50 value of 54.53 ug/mL[3]. |
Source |
Molecular Weight | 309.4 |
Formula | C20H23NO2 |
CAS No. | 5531-98-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (161.6 mM)
You can also refer to dose conversion for different animals. More
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Atherosperminine 5531-98-6 GPCR/G Protein Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience cAMP Calcium Channel AChR Parasite inhibit antiplasmodial Inhibitor pro-oxidant reductants Atherospermine trachealis inhibitor