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TOPProduct DescriptionPackaging & StorageSupporting FilesLibrary CustomizationLibrary Composition
TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
CDK
DNA/RNA Synthesis
Antibiotic
COX
NF-κB
EGFR
AChR
PI3K
Ras
Parasite
Adrenergic Receptor
HIV Protease
Calcium Channel
Dopamine Receptor
PDE
VEGFR
Dehydrogenase
Epigenetic Reader Domain
Potassium Channel
Histamine Receptor
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
Antifungal
Phosphatase
JAK
mTOR
Virus Protease
Src
p38 MAPK
SARS-CoV
Akt
FLT
ERK
Microtubule Associated
PARP
Cholinesterase (ChE)
Reactive Oxygen Species
TRP/TRPV Channel
PDGFR
Influenza Virus
Topoisomerase
iGluR
FGFR
PKC
Wnt/beta-catenin
STAT
TNF
Raf
Prostaglandin Receptor
HCV Protease
GSK-3
Bcl-2 Family
c-Kit
c-Met/HGFR
GABA Receptor
Monoamine Oxidase
Proteasome
RAAS
MAO
Caspase
MMP
NO Synthase
Bcr-Abl
Lipoxygenase
ALK
Ferroptosis
TGF-beta/Smad
HSP
NMDAR
Adenosine Receptor
MAPK
Phospholipase
DUB
Transferase
GluR
Histone Demethylase
Interleukin
GPCR
JNK
Aurora Kinase
E1/E2/E3 Enzyme
Beta Amyloid
Tyrosinase
Kras
PPAR
ROCK
Tyrosine Kinases
Serine Protease
Drug Metabolite
Anti-infection
HIF/HIF Prolyl-Hydroxylase
Casein Kinase
Integrin
AMPK
ATPase
PKA
Serotonin Transporter
Mitochondrial Metabolism
IL Receptor
Reductase
CCR
IκB/IKK
MEK
Serine/threonin kinase
Reverse Transcriptase
Carbonic Anhydrase
HSV
MDM-2/p53
Angiotensin-converting Enzyme (ACE)
Antiviral
Mitophagy
Nucleoside Antimetabolite/Analog
Cysteine Protease
Androgen Receptor
HBV
Glucosidase
Sirtuin
Estrogen Receptor/ERR
IGF-1R
Histone Acetyltransferase
Antioxidant
c-RET
Proton pump
DNA-PK
RIP kinase
ROS
CXCR
S6 Kinase
TAM Receptor
Norepinephrine
Acyltransferase
TLR
P-gp
HIF
Estrogen/progestogen Receptor
LPL Receptor
Leukotriene Receptor
Gamma-secretase
P2X Receptor
CaMK
c-Fms
FAK
NOS
FAAH
Opioid Receptor
Trk receptor
ATM/ATR
NADPH
DPP-4
Cannabinoid Receptor
NOD-like Receptor (NLR)
HER
Immunology/Inflammation related
Hedgehog/Smoothened
PLK
Neurokinin receptor
Syk
Glucocorticoid Receptor
Chk
p53
DYRK
Pim
Fatty Acid Synthase
NOD
HMG-CoA Reductase
Endothelin Receptor
DNA Methyltransferase
Kinesin
Chloride channel
PERK
IDO
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
Smo
transporter
Nrf2
Glutathione Peroxidase
SGLT
Hydroxylase
IRAK
PD-1/PD-L1
LTR
Rho
MAGL
LRRK2
PDK
Sigma receptor
ROS Kinase
P2Y Receptor
Lipase
Aryl Hydrocarbon Receptor
BTK
PAK
Thrombin
DHFR
Factor Xa
Isocitrate Dehydrogenase (IDH)
Xanthine Oxidase
PGE Synthase
S1P Receptor
Mdm2
YAP
BACE
c-Myc
Glutaminase
Myosin
cAMP
Retinoid Receptor
MRP
Cholecystokinin Receptor
IAP
OX Receptor
Epoxide Hydrolase
PI4K
Amino Acids and Derivatives
Glucokinase
IRE1
Stearoyl-CoA Desaturase (SCD)
Beta-Secretase
LPA Receptor
Complement System
Antifolate
CSF-1R
Aminopeptidase
Ephrin Receptor
ribosome
GTPase
Monoamine Transporter
Neuropeptide Y Receptor
Telomerase
OXPHOS
RSV
Aromatase
AhR
Monocarboxylate transporter
Ligands for Target Protein for PROTAC
DNA
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Tie-2
ABC Transporter
Lipid
PAI-1
GST
ADC Cytotoxin
MicroRNA
PAFR
Vasopressin Receptor
BCRP
Acetyl-CoA Carboxylase
Platelet aggregation
NADPH-oxidase
CFTR
MLK
Dynamin
MIF
DNA gyrase
Bradykinin Receptor
MNK
Survivin
Neprilysin
Melanocortin Receptor
CRM1
Na+/Ca2+ Exchanger
GNRH Receptor
Neurotensin Receptor
LIM Kinase
PYK2
NAMPT
FLAP
GRK
Molecular Glues
Wee1
OAT
Porcupine
STING
Methionine Adenosyltransferase (MAT)
SGK
MyD88
Necroptosis
SIK
UGT
LDL
Glucagon Receptor
Phosphorylase
GlyT
PAD
ATP Citrate Lyase
ASK
CRFR
Pyroptosis
Carboxypeptidase
APC/C
p97
Adenylyl Cyclase
Bcl-6
Prolyl Endopeptidase (PREP)
DNA Alkylation
PTEN
cGAS
GPX
Ligand for E3 Ligase
CGRP Receptor
DAPK
IKZF
ROR
MTP
IFNAR
Progesterone Receptor
Melatonin Receptor
AAK1
Arp2/3 Complex
Guanylate cyclase
MELK
Protease
Aquaporin
Gap Junction Protein
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
NEDD8
DprE1
Succinate Receptor 1 (SUCNR1)
DNA Alkylator/Crosslinker
CETP
Galectin
CaSR
ATG
FXR
NR4A
Amylase
MTH1
MT Receptor
Bombesin Receptor
CD73
Decarboxylase
Hippo pathway
KLF
CRISPR/Cas9
Oxytocin Receptor
Adenosine Deaminase
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
ASBT
Arrestin
TOPK
VDAC
LDLR
AAK1 (AP2 associated kinase 1)
Hexokinase
HCN Channel
ACK1
p62
FKBP
Imidazoline Receptor
Apelin receptor
CAT
Transaminase
Arginase
Factor VIIa
ASCT
Hck
Liver X Receptor
Endonuclease
Haspin Kinase
Na-K-Cl cotransporter
Somatostatin
KSP
Cadherin
GPCR19
AIM2
TSH Receptor
HuR
GHSR
FOXO
PKM
PGK1
GSNOR
NUDIX hydrolase
EBI2/GPR183
Y Box Binding Protein 1
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
RANKL/RANK
Annexin A
Neuropeptide FF Receptor
FABP
Integrase
Transketolase
hCE
Vitamin
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Photosensitizer
Stemness kinase
Photosystem (PS)
Adiponectin Receptor
Fas/FasL
PACAP
Anion Exchanger
PROTAC Linker
Thioredoxin
glycosidase
Mucin
Target Protein Ligand-Linker Conjugate
Huntingtin
PSMA
Glutathione reductase
MRGPR
Early 2 Factor (E2F)
Urea Transporter
CPT
CD74
GluCls
NEDD4-1
Cuproptosis
REV-ERB
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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