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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
AChR
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
Potassium Channel
Cytochromes P450
ROS
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
HDAC
ERK
Antifungal
Phosphatase
Akt
mTOR
JAK
Virus Protease
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
STAT
Influenza Virus
Wnt/beta-catenin
TNF
iGluR
PDGFR
PARP
Reactive Oxygen Species
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
FGFR
GSK-3
PKC
Caspase
Interleukin
Raf
Bcl-2 Family
NO Synthase
HCV Protease
c-Kit
Monoamine Oxidase
GABA Receptor
MMP
c-Met/HGFR
Proteasome
RAAS
MAO
Lipoxygenase
JNK
Ferroptosis
Bcr-Abl
TGF-beta/Smad
ALK
MAPK
HSP
Phospholipase
Transferase
Adenosine Receptor
NMDAR
E1/E2/E3 Enzyme
DUB
GluR
Histone Demethylase
Drug Metabolite
PPAR
Tyrosinase
Beta Amyloid
Aurora Kinase
GPCR
Serine Protease
Integrin
ROCK
Kras
HIF/HIF Prolyl-Hydroxylase
Serotonin Transporter
Tyrosine Kinases
Casein Kinase
Anti-infection
Reductase
PKA
AMPK
CCR
MDM-2/p53
MEK
Mitochondrial Metabolism
IL Receptor
IκB/IKK
Serine/threonin kinase
ATPase
HSV
Carbonic Anhydrase
Reverse Transcriptase
Angiotensin-converting Enzyme (ACE)
Nucleoside Antimetabolite/Analog
P-gp
HBV
IGF-1R
Antiviral
Androgen Receptor
Mitophagy
Estrogen Receptor/ERR
Sirtuin
Cysteine Protease
CXCR
TLR
Glucosidase
Histone Acetyltransferase
RIP kinase
Antioxidant
Proton pump
Acyltransferase
c-RET
glycosidase
CaMK
TAM Receptor
FAK
S6 Kinase
DNA-PK
Leukotriene Receptor
Norepinephrine
NOD-like Receptor (NLR)
HIF
LPL Receptor
P2X Receptor
Gamma-secretase
Trk receptor
c-Fms
NOS
Estrogen/progestogen Receptor
PERK
Cannabinoid Receptor
ATM/ATR
FAAH
Hedgehog/Smoothened
Opioid Receptor
Nrf2
NADPH
Immunology/Inflammation related
Chk
HER
Fatty Acid Synthase
Kinesin
DPP-4
PLK
Syk
Neurokinin receptor
IDO
Glucocorticoid Receptor
Indoleamine 2,3-Dioxygenase (IDO)
p53
Pim
DYRK
NOD
Lipase
HMG-CoA Reductase
PD-1/PD-L1
Endothelin Receptor
Chloride channel
Glutathione Peroxidase
transporter
PDK
Antifection
DNA Methyltransferase
Xanthine Oxidase
SGLT
Smo
Hydroxylase
Aryl Hydrocarbon Receptor
IRAK
Thrombin
LTR
MAGL
LRRK2
Rho
Sigma receptor
ROS Kinase
YAP
c-Myc
BTK
Isocitrate Dehydrogenase (IDH)
PAK
Glutaminase
P2Y Receptor
Stearoyl-CoA Desaturase (SCD)
Factor Xa
PGE Synthase
S1P Receptor
DHFR
IAP
Retinoid Receptor
Mdm2
cAMP
Amino Acids and Derivatives
Epoxide Hydrolase
BACE
MRP
Antifolate
OX Receptor
Aminopeptidase
PI4K
Cholecystokinin Receptor
Myosin
Beta-Secretase
IRE1
LPA Receptor
Glucokinase
Complement System
Monoamine Transporter
Monocarboxylate transporter
OXPHOS
Neuropeptide Y Receptor
Ephrin Receptor
RSV
CSF-1R
ribosome
Telomerase
Lipid
GTPase
PAI-1
Aromatase
AhR
DNA
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Ligands for Target Protein for PROTAC
ABC Transporter
MLK
GST
CFTR
Adenylate cyclase
Dynamin
PAFR
Tie-2
ADC Cytotoxin
STING
Acetyl-CoA Carboxylase
NADPH-oxidase
Necroptosis
GRK
Vasopressin Receptor
Platelet aggregation
MicroRNA
DNA gyrase
Bradykinin Receptor
Pyroptosis
Molecular Glues
Melanocortin Receptor
MIF
OAT
MNK
Neprilysin
Porcupine
MyD88
SGK
Na+/Ca2+ Exchanger
GNRH Receptor
NAMPT
Carboxypeptidase
CRM1
Neurotensin Receptor
PYK2
UGT
GlyT
Wee1
Methionine Adenosyltransferase (MAT)
p97
LIM Kinase
Glucagon Receptor
FLAP
ATP Citrate Lyase
Prolyl Endopeptidase (PREP)
CGRP Receptor
Phosphorylase
CRFR
Gap Junction Protein
PAD
ASK
DAPK
SIK
IKZF
APC/C
MTP
PROTACs
cGAS
LDL
PTEN
GPX
IFNAR
Bcl-6
Arp2/3 Complex
Ligands for E3 Ligase
Protease
LDLR
DNA Alkylation
Hippo pathway
DNA Alkylator/Crosslinker
Arrestin
Melatonin Receptor
Guanylate cyclase
Progesterone Receptor
MELK
Aquaporin
ROR
AAK1
NEDD8
ATG
NR4A
CD73
MALT
DprE1
FXR
Amylase
CETP
MT Receptor
Bombesin Receptor
CaSR
Liver X Receptor
HCN Channel
Oxytocin Receptor
Galectin
MTH1
KLF
BMI-1
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
Succinate Receptor 1 (SUCNR1)
Decarboxylase
FOXO
Adenosine Deaminase
CD38
VDAC
Vitamin
p62
CRISPR/Cas9
FKBP
Advanced Glycation End Products
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
ACK1
Imidazoline Receptor
ASBT
PKM
Hexokinase
Orphan Receptor
NPC1L1
TOPK
Factor VIIa
Endonuclease
PROTAC Linker
TSH Receptor
FABP
KSP
Cadherin
Hck
HuR
CAT
Arginase
ASCT
AIM2
GHSR
Transaminase
Somatostatin
Apelin receptor
Haspin Kinase
GPCR19
Ferroportin
PGK1
Transketolase
Huntingtin
NUDIX hydrolase
RANKL/RANK
Annexin A
PSMA
hCE
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
gp120/CD4
Photosensitizer
Glutaminyl Cyclase
Urea Transporter
Kisspeptin
Neuropeptide FF Receptor
Integrase
PARG（Poly(ADP-ribose) Glycohydrolase）
FOXO3
Drug-Linker Conjugates for ADC
stilbene oxidase
VDA
N-Acetylglucosaminyltransferase
Target Protein Ligand-Linker Conjugates
LAG-3
Photosystem (PS)
Adiponectin Receptor
Anion Exchanger
E3 Ligase Ligand-Linker Conjugates
CD74
RAR/RXR
Neuropeptide W
PACAP
MRGPR
GluCls
Piezo Channel
Procollagen C Proteinase
Cell wall
OCT
Stemness kinase
Fas/FasL
Early 2 Factor (E2F)
LHRH
CPT
REV-ERB
Mucin
Cuproptosis
Glyoxalase
Lysosomal Autophagy
NEDD4-1
Fer/FerT kinase
Tight Junction Protein
Taste receptor
Aconitase
Thioredoxin
Glutathione reductase
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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