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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7147 | Valbenazine | NBI-98854 | Monoamine Transporter |
Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia. | |||
T3280 | Clodronate disodium tetrahydrate | clodronic acid disodium tetrahydrate,Disodium clodronate tetrahydrate,Clastoban,Clodronate disodium | IL Receptor , TNF |
Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification. | |||
T7563 | NBI-98782 | (+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ | Monoamine Transporter |
NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM) | |||
T23409 | FM4-64 | SynaptoRedTM C2 | Others |
FM4-64 (SynaptoRedTM C2) is a styryl dye that stains stably but does not fluoresce in aqueous solution.FM4-64 does not passively diffuse into the plasma membrane bilayer and must be actively transported across the membra... | |||
TP1429 | VSV-G Peptide acetate(103425-05-4 free base) | VSV-G Peptide | Others |
VSV-G Peptide acetate(103425-05-4 free base) is a 11 amino acid peptide derived from the Vesicular Stomatitis viral glycoprotein. | |||
T13134 | (+)-Tetrabenazine | (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ | Monoamine Transporter |
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. | |||
T22486 | Vesamicol hydrochloride | (±)-AH5183 hydrochloride | AChR |
Vesamicol hydrochloride ((±)-AH5183 hydrochloride) is a acetylcholine transport inhibitor. | |||
T7651 | Rose Bengal sodium | Rose Bengal | Influenza Virus , Monoamine Transporter |
Rose Bengal sodium is a potent inhibitor of VGlut and vesicular monoamine transporter (VMAT) (Ki of 19 and 64 nM for VGlut andVMAT, respectively) | |||
T3534 | Tetrabenazine Racemate | Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE | Monoamine Transporter |
Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been ... | |||
T77549 | Nurr1 agonist 2 | Others | |
Nurr1 agonist 2 is a Nurr1 agonist with an EC50 value of 0.07 μM. Nurr1 agonist 2 increases the mRNA expression of the Nurr1-regulated genes tyrosine hydroxylase (TH) and vesicular amino acid transporter 2 (VMAT2). Nurr1... | |||
T22781L | FFN 511 hydrochloride | FFN 511 hydrochloride(1004548-96-2 Free base) | |
FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitters (FFNs) targeting neuronal vesicular monoamine transporter 2 (VMA T2).FFN 511 hydrochloride inhibits the binding of 5-hydroxytryptamine to VMA T2-containing ... | |||
T0313 | Evans blue | Direct Blue 53,C.I. 23860 | GluR |
Evans blue (C.I. 23860) is an azo dye, inhibits L-glutamate uptake via the membrane-bound excitatory amino acid transporter (EAAT). | |||
T36949 | Niaprazine | 5-HT Receptor , Adrenergic Receptor , Histamine Receptor | |
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff... | |||
T25750 | Lobelane Hydrochloride | ||
Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor. | |||
T31791 | FFN246 HCl | FFN 246,FFN246 hydrochloride,FFN246,FFN-246 | |
FFN246 is a fluorescent substrate for both the serotonin transporter and the vesicular monoamine transporter 2 (VMAT2). | |||
T24941 | VMAT2-IN-I HCl | VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride | |
VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A. | |||
T31790 | FFN200 dihydrochloride | FFN200 HCl,FFN200,FFN 200,FFN-200 | |
FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue. | |||
T12190 | Trans (2,3)-Dihydrotetrabenazine | (2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine | Others |
Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2). | |||
T70322 | Valbenazine dihydrochloride | ||
Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia. | |||
T22452 | Valbenazine tosylate | NBI-98854 | Monoamine Transporter |
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM). |