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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TN6848 | Piperonylic acid | 2H-1,3-benzodioxole-5-carboxylic acid | P450 |
Piperonylic acid (2H-1,3-benzodioxole-5-carboxylic acid) is a natural molecule bearing a methylenedioxy function that closely mimics the structure of trans-cinnamic acid. Piperonylic acid selectively inactivate the CYP73... | |||
T20189 | Benzoylphenylalanine | L-BPA,NSC118532,N-Benzoyl-L-phenylalanine,LBPA,NSC-118532,L BPA,NSC 118532 | Others |
Benzoylphenylalanine (LBPA) can be used as a photoaffinity peptide inactivator. | |||
T6S1894 | Linderane | P450 | |
1. Linderane was characterized as a mechanism-based inactivator of CYP2C9. | |||
T3677 | GSK2879552 | GSK2879552 2HCl | Histone Demethylase |
GSK2879552 is a selective, orally bioavailable, irreversible, mechanism-based inactivator of lysine-specific demethylase 1 (LSD1)/corepressor, with potential antineoplastic activity. | |||
T7539 | O6-Benzylguanine | Apoptosis , DNA Alkylation , DNA/RNA Synthesis | |
O6-Benzylguanine is a guanine analog with antineoplastic activity,and is a potent O6-alkylguanine DNA alkyltransferase (AGT) inactivator. | |||
T3776 | Rhapontigenin | Protigenin | P450 , Antibacterial , Antifungal |
Rhapontigenin (Protigenin) is a mechanism-based, selective inactivator of cytochrome P450 1A1 (IC50: 400 nM), an aryl hydrocarbon hydroxylase which activates polycyclic aromatic hydrocarbons that act as procarcinogens. R... | |||
T25217 | CDE-096 | ||
CDE-096 is a plasminogenactivator inhibitor-1 (PAI-1) inactivator. | |||
T71709 | MDL-72527 free base | ||
MDL-72527 free base is a polyamine oxidase inactivator. | |||
T63342 | Anti-TSWV agent 1 | ||
Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV). | |||
T24054 | F-amidine | ||
F-amidine is a bioavailable irreversible PAD4 inactivator. | |||
T26402 | A 1110U | A-1110U,A1110U | |
A 1110U is an inactivator of herpes simplex virus ribonucloetide reductases. | |||
T73530 | 2-PAT | ||
2-PAT, analogous to Rasagiline and Selegiline, functions as a reversible MAO-A inhibitor, exhibiting an IC50 of 0.721 µM, and acts as an inactivator of MAO-B with an IC50 value of 14.6 µM. This compound shows promise for... |