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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP2032 | Des-Gln14-Ghrelin | des-Gln14-Ghrelin (rat) | |
An endogenous ligand for the ghrelin receptor (GHS-R1a), produced by alternative splicing of the rat ghrelin gene. Potently induces Ca2+ release in cells expressing ghrelin receptors (EC50 = 2.4 nM) and stimulates GH rel... | |||
T40234 | Ghrelin receptor full agonist-2 | ||
Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist. | |||
TP2241 | [Des-octanoyl]-Ghrelin (human) | Others | |
[Des-octanoyl]-Ghrelin (human) is a Non-acylated, major circulating isoform of ghrelin. | |||
TP2242 | [Des-octanoyl]-Ghrelin (rat) | Others | |
[Des-octanoyl]-Ghrelin (rat) is a Non-acylated, major circulating isoform of ghrelin. | |||
T75928 | Des-Gln14-Ghrelin TFA | ||
Des-Gln14-Ghrelin TFA serves as a potent endogenous ligand for the growth hormone secretagogue receptor, effectively inducing increases in intracellular calcium levels ([Ca2+]i) in CHO-GHSR62 cells with an EC50 of 2.4 nM... | |||
T2O2721 | L-Cysteine | Thioserine,cysteine,L-(+)-Cysteine | Endogenous Metabolite |
L-Cysteine (L-(+)-Cysteine) is a non-essential sulfur-containing amino acid in humans. L-Cysteine is important for protein synthesis, detoxification, and diverse metabolic functions. Found in beta-keratin, the main prote... | |||
T80006 | Emoghrelin | GHSR | |
Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1]. | |||
T10319 | Anamorelin | RC-1291,ONO-7643 | GHSR |
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). | |||
T16508 | PF-5190457 | PF-05190457 | GHSR |
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36). | |||
T7225 | AnaMorelin hydrochloride | RC-1291 hydrochloride,ONO-7643 hydrochloride | GHSR |
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay). | |||
T23543 | YIL 781 | GHSR | |
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM). YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion... | |||
TP1931L1 | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) | cholecystokinin |
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ... | |||
T8141 | L-Cysteine hydrochloride | L-Cysteine HCl | Others , Endogenous Metabolite |
L-Cysteine hydrochloride (L-Cysteine HCl) is a conditionally essential amino acid,L-Cysteine hydrochloride suppresses ghrelin and reduces appetite in rodents and humans | |||
TN5283 | L-Cysteine hydrochloride hydrate | L-Cysteine hydrochloride monohydrate | Others , Endogenous Metabolite |
L-Cysteine hydrochloride hydrate (L-Cysteine hydrochloride monohydrate) is a conditionally essential amino acid, which acts as a precursor for biologically active molecules such as hydrogen sulphide (H2S), taurine and gl... | |||
T10319L | Anamorelin Fumarate | ONO-7643 Fumarate,RC1291 Fumarate | Others |
Anamorelin Fumarate is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). | |||
T34281 | Relamorelin | BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131 | GHSR |
Relamorelin (RM-131), a selective and potent growth hormone-releasing peptide/growth hormone secretagogue receptor (GHSR) agonist, is a potent growth hormone-releasing peptide mimetic with a high affinity for the GHS-1a ... | |||
T22898 | L-692585 | L-692,585 | Others |
ghrelin receptor (GHS-R1a) agonist | |||
T27443 | GSK 894281 | GSK894281,GSK-894281 | |
GSK 894281 is a ghrelin receptor agonist. It may produces myocardial degeneration/necrosis in rats. | |||
T27451 | GSK1614343 | GSK-1614343,GSK 1614343 | |
GSK1614343 is an antagonist of ghrelin receptor. | |||
T23413 | Tabimorelin hemifumarate | Others | |
orally active ghrelin receptor (GHS-R1a) agonist |